FAIRMol

TC268

Pose ID 5356 Compound 749 Pose 2038

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good fit quality (FQ -2.26) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (43.1 kcal/mol) ✗ Low LE (-0.194 kcal/mol/HA) ✗ Geometry warnings ℹ SASA not computed
Score
-13.025
kcal/mol
LE
-0.194
kcal/mol/HA
Fit Quality
-2.26
FQ (Leeson)
HAC
67
heavy atoms
MW
939
Da
LogP
5.54
cLogP
Strain ΔE
43.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: acceptable
Geometry reliability: low
Reason: geometry warning, clashes, strain 43.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 3 Clashes 18 Severe clashes 4
Final rank63.95618221165056Score-13.0253
Inter norm-0.285993Intra norm0.0908728
Top1000noExcludedyes
Contacts16H-bonds5
Artifact reasonexcluded; geometry warning; 21 clashes; 4 protein clashes
ResiduesA:ARG97;A:ASN58;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:PRO93;A:SER86;A:THR54;A:THR83;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap12Native recall0.60
Jaccard0.50RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
966 7.924960003015377 -0.230019 -10.6205 5 16 0 0.00 0.00 - no Open
971 8.622410915467011 -0.262052 -14.6976 8 18 0 0.00 0.00 - no Open
963 8.668732509650429 -0.262062 -19.966 11 16 0 0.00 0.00 - no Open
973 9.829918695358124 -0.311862 -14.6976 8 15 0 0.00 0.00 - no Open
2033 9.859658197352427 -0.403028 -4.90992 6 21 15 0.75 0.40 - no Open
2031 11.031232536328456 -0.495192 -21.8006 7 19 12 0.60 0.20 - no Open
2040 10.267799486580678 -0.49344 -21.1745 2 25 18 0.90 0.00 - yes Open
964 10.408910837040514 -0.237622 -10.2971 7 20 0 0.00 0.00 - yes Open
2036 10.480489535050769 -0.388256 -23.9808 4 20 14 0.70 0.00 - yes Open
972 12.733866709987094 -0.219659 -8.63375 7 17 0 0.00 0.00 - yes Open
2037 13.398149860971646 -0.32272 -13.9885 7 19 13 0.65 0.20 - yes Open
2039 15.008648071697358 -0.387667 -18.7564 9 23 16 0.80 0.20 - yes Open
2029 57.916787006582524 -0.34104 -18.6838 6 21 15 0.75 0.20 - yes Open
2030 58.04003634870706 -0.410412 -21.6919 6 23 18 0.90 0.40 - yes Open
968 58.1921685393656 -0.251457 -6.81459 7 18 0 0.00 0.00 - yes Open
2034 58.308985218766225 -0.395443 -12.0484 3 20 14 0.70 0.40 - yes Open
967 58.3695528382883 -0.298086 -10.1592 7 21 0 0.00 0.00 - yes Open
969 58.76365490072506 -0.351447 -19.3528 11 22 0 0.00 0.00 - yes Open
2035 59.2106178894737 -0.39712 -19.9826 5 18 11 0.55 0.20 - yes Open
962 60.09819276727043 -0.248705 -24.6375 7 16 0 0.00 0.00 - yes Open
2032 61.28527412652558 -0.43473 -20.7284 6 17 11 0.55 0.20 - yes Open
965 62.22827217570115 -0.341314 -18.1706 9 22 0 0.00 0.00 - yes Open
970 63.08438541607137 -0.22874 -12.9469 7 19 0 0.00 0.00 - yes Open
2038 63.95618221165056 -0.285993 -13.0253 5 16 12 0.60 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -13.025kcal/mol
Ligand efficiency (LE) -0.1944kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -2.256
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 67HA

Physicochemical properties

Molecular weight 939.1Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.54
Lipinski: ≤ 5
Rotatable bonds 14

Conformational strain (MMFF94s)

Strain energy (ΔE) 43.12kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 193.39kcal/mol
Minimised FF energy 150.27kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.