FAIRMol

TC71

Pose ID 5308 Compound 253 Pose 1990

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.626 kcal/mol/HA) ✓ Good fit quality (FQ -6.26) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (43.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.273
kcal/mol
LE
-0.626
kcal/mol/HA
Fit Quality
-6.26
FQ (Leeson)
HAC
34
heavy atoms
MW
483
Da
LogP
5.37
cLogP
Strain ΔE
43.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 43.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 1 Clashes 8 Severe clashes 2
Final rank57.10592140478446Score-21.2727
Inter norm-0.655981Intra norm0.030314
Top1000noExcludedyes
Contacts16H-bonds3
Artifact reasonexcluded; geometry warning; 14 clashes; 2 protein clashes
ResiduesA:ALA32;A:ASN58;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:THR54;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap15Native recall0.75
Jaccard0.71RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1905 5.104866815228245 -0.710523 -26.0124 2 20 0 0.00 0.00 - no Open
1907 6.175050330553141 -0.635334 -20.1282 1 20 0 0.00 0.00 - no Open
1987 6.493443960901055 -0.667066 -23.1803 3 19 18 0.90 0.20 - no Open
1909 7.101960946007024 -0.801899 -30.7153 8 22 0 0.00 0.00 - no Open
1993 7.441618172275733 -0.683262 -20.4478 3 18 18 0.90 0.00 - no Open
1988 7.755716690108713 -0.790421 -25.5478 2 17 17 0.85 0.20 - yes Open
1906 55.04519385134802 -0.670851 -23.0018 3 18 0 0.00 0.00 - yes Open
1991 56.49799754134236 -0.645669 -22.8663 4 14 10 0.50 0.20 - yes Open
1910 56.752469651210745 -0.629057 -21.7106 9 21 0 0.00 0.00 - yes Open
1989 56.92236331963167 -0.679926 -24.5927 3 20 18 0.90 0.20 - yes Open
1990 57.10592140478446 -0.655981 -21.2727 3 16 15 0.75 0.00 - yes Current
1911 57.26577548493912 -0.580617 -21.0767 8 16 0 0.00 0.00 - yes Open
1908 58.39041328417018 -0.612291 -22.19 6 17 0 0.00 0.00 - yes Open
1992 58.52225989130012 -0.647248 -23.4862 3 17 16 0.80 0.00 - yes Open
1986 58.95174772421978 -0.812852 -25.8237 4 16 11 0.55 0.20 - yes Open
1904 60.214299205472514 -0.626782 -22.1073 9 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.273kcal/mol
Ligand efficiency (LE) -0.6257kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.260
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 482.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.37
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 43.10kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 73.36kcal/mol
Minimised FF energy 30.26kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.