FAIRMol

Z44355105

Pose ID 52822 Compound 3333 Pose 2966

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.214 kcal/mol/HA) ✓ Good fit quality (FQ -10.72) ✓ Strong H-bond network (10 bonds) ✗ High strain energy (12.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-27.929
kcal/mol
LE
-1.214
kcal/mol/HA
Fit Quality
-10.72
FQ (Leeson)
HAC
23
heavy atoms
MW
344
Da
LogP
3.20
cLogP
Strain ΔE
12.1 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 10 Hydrophobic 12 π–π 3 Clashes 10 Severe clashes 0
Final rank4.043722053723348Score-27.9292
Inter norm-1.07128Intra norm-0.143028
Top1000noExcludedno
Contacts17H-bonds10
Artifact reasongeometry warning; 9 clashes; 10 protein contact clashes; moderate strain Δ 13.7
ResiduesA:ARG137;A:ARG141;A:ASN103;A:HIS102;A:MET98;A:TYR94;B:ARG113;B:ASP10;B:CYS69;B:GLY70;B:GLY72;B:GLY74;B:HIS11;B:ILE73;B:PRO12;B:SER71;B:TYR46

Protein summary

305 residues
Protein targetT21Atoms4646
Residues305Chains2
Residue summaryARG:576; ILE:532; VAL:512; GLU:420; ALA:360; PHE:240; HIS:238; LYS:220; THR:210; LEU:190; PRO:168; TYR:168; GLY:154; SER:154; ASP:144; ASN:112

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3K7OContacts14
PoseOpen native poseH-bonds16
IFP residuesA:ARG137; A:ARG141; A:ASN103; A:HIS102; A:HIS138; B:ASP10; B:CYS69; B:GLY70; B:GLY74; B:HIS11; B:ILE73; B:PRO12; B:SER71; B:TYR46
Current overlap13Native recall0.93
Jaccard0.72RMSD-
H-bond strict6Strict recall0.50
H-bond same residue+role5Role recall0.56
H-bond same residue5Residue recall0.62

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2801 3.677793333105896 -0.819958 -19.7281 5 10 0 0.00 0.00 - no Open
2966 4.043722053723348 -1.07128 -27.9292 10 17 13 0.93 0.56 - no Current
2802 4.094901877936572 -0.747803 -20.2781 3 9 0 0.00 0.00 - no Open
2965 4.7088080297849535 -0.947034 -22.9296 10 16 14 1.00 0.56 - no Open
2800 7.5215465968494915 -0.733813 -18.182 4 10 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -27.929kcal/mol
Ligand efficiency (LE) -1.2143kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -10.717
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 344.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.20
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 12.07kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 54.87kcal/mol
Minimised FF energy 42.80kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.