FAIRMol

Z56833421

Pose ID 52467 Compound 1647 Pose 2611

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-1.074 kcal/mol/HA) ✓ Good fit quality (FQ -9.89) ✓ Strong H-bond network (13 bonds) ✗ Very high strain energy (30.4 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-27.921
kcal/mol
LE
-1.074
kcal/mol/HA
Fit Quality
-9.89
FQ (Leeson)
HAC
26
heavy atoms
MW
378
Da
LogP
0.79
cLogP
Strain ΔE
30.4 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 13 Hydrophobic 5 π–π 1 Clashes 9 Severe clashes 0
Final rank6.093663981989673Score-27.9214
Inter norm-1.04611Intra norm-0.0277892
Top1000noExcludedno
Contacts17H-bonds13
Artifact reasongeometry warning; 7 clashes; 9 protein contact clashes; high strain Δ 56.3
ResiduesA:ARG137;A:ARG141;A:ASN103;A:HIS102;A:MET98;A:TYR94;B:ARG113;B:ASP10;B:CYS69;B:GLY70;B:GLY72;B:GLY74;B:HIS11;B:ILE73;B:PRO12;B:SER71;B:TYR46

Protein summary

305 residues
Protein targetT21Atoms4646
Residues305Chains2
Residue summaryARG:576; ILE:532; VAL:512; GLU:420; ALA:360; PHE:240; HIS:238; LYS:220; THR:210; LEU:190; PRO:168; TYR:168; GLY:154; SER:154; ASP:144; ASN:112

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3K7OContacts14
PoseOpen native poseH-bonds16
IFP residuesA:ARG137; A:ARG141; A:ASN103; A:HIS102; A:HIS138; B:ASP10; B:CYS69; B:GLY70; B:GLY74; B:HIS11; B:ILE73; B:PRO12; B:SER71; B:TYR46
Current overlap13Native recall0.93
Jaccard0.72RMSD-
H-bond strict4Strict recall0.33
H-bond same residue+role4Role recall0.44
H-bond same residue4Residue recall0.50

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2200 3.5036189774168602 -0.909604 -21.449 5 16 0 0.00 0.00 - no Open
3541 3.603392263402044 -0.761299 -17.4524 5 15 0 0.00 0.00 - no Open
2196 3.881262193448731 -1.06544 -27.514 7 16 0 0.00 0.00 - no Open
2199 4.195608556104308 -0.949774 -22.9721 7 14 0 0.00 0.00 - no Open
3543 4.366012830636955 -0.739141 -17.5495 7 13 0 0.00 0.00 - no Open
1942 4.4813218657358105 -1.19127 -27.2964 11 15 0 0.00 0.00 - no Open
2204 4.8782940730045095 -0.864456 -24.9424 5 16 0 0.00 0.00 - no Open
2195 4.93734756640286 -0.997851 -23.7203 9 16 0 0.00 0.00 - no Open
3537 4.979313511661527 -0.8042 -18.3974 5 12 0 0.00 0.00 - no Open
1947 5.320563734704506 -1.23255 -30.9792 10 15 0 0.00 0.00 - no Open
2080 5.43529727290073 -0.899153 -21.0407 13 17 0 0.00 0.00 - no Open
2611 6.093663981989673 -1.04611 -27.9214 13 17 13 0.93 0.44 - no Current
2364 6.2295396317531875 -0.975955 -23.742 7 14 0 0.00 0.00 - no Open
3542 6.4806037186103636 -0.771504 -16.2998 9 14 0 0.00 0.00 - no Open
2203 6.898506052662953 -1.00733 -23.6968 9 16 0 0.00 0.00 - no Open
1941 4.929374925320752 -1.30893 -33.2869 8 14 0 0.00 0.00 - yes Open
1943 5.555768727869188 -1.23287 -34.608 11 11 0 0.00 0.00 - yes Open
2197 5.700320088194233 -0.927718 -25.4303 4 14 0 0.00 0.00 - yes Open
2078 5.72617750474478 -1.01408 -22.2016 11 17 0 0.00 0.00 - yes Open
2082 6.707896967070407 -0.95306 -24.6346 12 18 0 0.00 0.00 - yes Open
2355 6.764994635319981 -0.905288 -18.1166 8 10 0 0.00 0.00 - yes Open
1949 6.9293501710947 -1.26455 -33.6303 9 12 0 0.00 0.00 - yes Open
1946 7.2341253755488495 -1.14676 -31.8341 11 16 0 0.00 0.00 - yes Open
2077 7.236027629908628 -0.951395 -27.6673 9 16 0 0.00 0.00 - yes Open
2363 7.35940865034636 -0.80857 -25.4456 9 10 0 0.00 0.00 - yes Open
2201 7.420394837931003 -0.952816 -27.7319 8 19 0 0.00 0.00 - yes Open
2083 7.4364677837408735 -1.04357 -29.9915 16 15 0 0.00 0.00 - yes Open
2619 7.47192955099834 -0.892317 -18.9751 9 12 10 0.71 0.44 - yes Open
2079 7.557973534059099 -1.04788 -29.5821 8 17 0 0.00 0.00 - yes Open
2356 7.831486111797295 -0.989873 -21.3665 9 14 0 0.00 0.00 - yes Open
2615 7.897952123744167 -0.947079 -23.2985 10 15 12 0.86 0.67 - yes Open
2357 7.980590544053714 -0.829523 -20.637 12 14 0 0.00 0.00 - yes Open
1945 8.190803097696365 -1.20616 -31.2214 10 12 0 0.00 0.00 - yes Open
1948 8.352754565848604 -1.395 -34.3545 16 11 0 0.00 0.00 - yes Open
2358 8.448303964044678 -0.783971 -19.3556 7 11 0 0.00 0.00 - yes Open
3539 8.452148263410667 -0.722552 -19.9782 5 13 0 0.00 0.00 - yes Open
2075 8.533512774415247 -1.07197 -20.1527 10 16 0 0.00 0.00 - yes Open
2610 8.560105549858074 -1.07884 -24.8429 11 15 12 0.86 0.44 - yes Open
2618 8.641412429057167 -0.925655 -26.227 12 17 13 0.93 0.67 - yes Open
2360 8.708859461467467 -0.821692 -18.9942 9 11 0 0.00 0.00 - yes Open
2616 8.779735936129157 -0.923269 -23.05 12 16 13 0.93 0.67 - yes Open
2202 8.906247037959892 -0.848173 -19.6083 11 14 0 0.00 0.00 - yes Open
2081 9.067324973435559 -1.14702 -29.589 14 14 0 0.00 0.00 - yes Open
2362 9.453217537638405 -0.924583 -20.1765 10 16 0 0.00 0.00 - yes Open
2613 9.692961274563716 -0.901154 -20.9216 14 14 13 0.93 0.78 - yes Open
3540 9.767383562808194 -0.808893 -21.9366 7 16 0 0.00 0.00 - yes Open
3536 9.902347763280268 -0.904088 -20.6734 8 14 0 0.00 0.00 - yes Open
2084 10.0029587700547 -1.09933 -26.5643 13 17 0 0.00 0.00 - yes Open
3538 10.23397027380129 -0.864932 -20.7495 9 13 0 0.00 0.00 - yes Open
1950 10.32260872090762 -1.47787 -38.8504 14 15 0 0.00 0.00 - yes Open
2361 10.397735414069864 -0.775763 -18.6675 13 12 0 0.00 0.00 - yes Open
2614 10.434216413583206 -0.970019 -23.8333 13 16 11 0.79 0.78 - yes Open
2076 10.495597177909964 -0.999051 -26.9445 9 17 0 0.00 0.00 - yes Open
1944 11.101108336459667 -0.993802 -24.1175 5 12 0 0.00 0.00 - yes Open
2612 12.012578235153534 -0.919665 -23.9389 14 15 12 0.86 0.78 - yes Open
2359 12.0919616081992 -1.08851 -28.813 14 16 0 0.00 0.00 - yes Open
2617 12.570897429512385 -0.931936 -19.1351 12 16 13 0.93 0.44 - yes Open
2198 15.161449616086365 -0.871529 -21.2385 9 13 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -27.921kcal/mol
Ligand efficiency (LE) -1.0739kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -9.894
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 378.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.79
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 30.41kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 116.98kcal/mol
Minimised FF energy 86.58kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.