FAIRMol

Z44844875

Pose ID 52459 Compound 2331 Pose 2603

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.542 kcal/mol/HA) ✓ Good fit quality (FQ -5.28) ✓ Strong H-bond network (9 bonds) ✗ High strain energy (19.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-16.793
kcal/mol
LE
-0.542
kcal/mol/HA
Fit Quality
-5.28
FQ (Leeson)
HAC
31
heavy atoms
MW
418
Da
LogP
4.87
cLogP
Strain ΔE
19.1 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 9 Hydrophobic 4 π–π 3 Clashes 6 Severe clashes 0 ⚠ Hydrophobic exposure 52%
⚠️Partial hydrophobic solvent exposure
52% of hydrophobic surface appears solvent-exposed (13/25 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 25 Buried (contacted) 12 Exposed 13 LogP 4.87 H-bonds 9
Exposed fragments: phenyl (6/6 atoms exposed)aliphatic chain/group (7 atoms exposed)
Final rank4.970431183587568Score-16.7932
Inter norm-0.587359Intra norm0.0456417
Top1000noExcludedno
Contacts16H-bonds9
Artifact reasongeometry warning; 14 clashes; 6 protein contact clashes; high strain Δ 23.1
ResiduesA:ARG137;A:ARG141;A:ASN103;A:HIS102;A:MET98;A:TYR94;B:ARG113;B:ASP10;B:CYS69;B:GLY70;B:GLY74;B:HIS11;B:ILE73;B:PRO12;B:SER71;B:TYR46

Protein summary

305 residues
Protein targetT21Atoms4646
Residues305Chains2
Residue summaryARG:576; ILE:532; VAL:512; GLU:420; ALA:360; PHE:240; HIS:238; LYS:220; THR:210; LEU:190; PRO:168; TYR:168; GLY:154; SER:154; ASP:144; ASN:112

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3K7OContacts14
PoseOpen native poseH-bonds16
IFP residuesA:ARG137; A:ARG141; A:ASN103; A:HIS102; A:HIS138; B:ASP10; B:CYS69; B:GLY70; B:GLY74; B:HIS11; B:ILE73; B:PRO12; B:SER71; B:TYR46
Current overlap13Native recall0.93
Jaccard0.76RMSD-
H-bond strict5Strict recall0.42
H-bond same residue+role5Role recall0.56
H-bond same residue4Residue recall0.50

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2603 4.970431183587568 -0.587359 -16.7932 9 16 13 0.93 0.56 - no Current
2459 5.283698177054297 -0.568492 -19.7534 6 9 0 0.00 0.00 - no Open
2064 7.323797290416142 -0.810191 -30.4895 9 18 0 0.00 0.00 - no Open
2060 7.4413794267973445 -0.805549 -24.7691 10 19 0 0.00 0.00 - no Open
2598 6.057633307738709 -0.76343 -21.2631 5 17 13 0.93 0.44 - yes Open
2065 6.480752843876996 -0.798298 -24.4765 10 17 0 0.00 0.00 - yes Open
2602 6.779895029604055 -0.720747 -22.7613 8 17 13 0.93 0.56 - yes Open
2461 6.906583323998046 -0.577292 -18.023 6 12 0 0.00 0.00 - yes Open
2462 6.955028032851434 -0.49098 -15.2632 4 11 0 0.00 0.00 - yes Open
2601 7.153191856958005 -0.605953 -19.4329 7 15 12 0.86 0.56 - yes Open
2599 7.307388460417495 -0.650187 -21.9386 10 16 12 0.86 0.56 - yes Open
2463 7.593777531084623 -0.462227 -13.502 3 10 0 0.00 0.00 - yes Open
2062 7.623365461212505 -0.689706 -20.3921 6 17 0 0.00 0.00 - yes Open
2063 8.06591193248797 -0.812272 -28.593 10 16 0 0.00 0.00 - yes Open
2600 8.846237669105472 -0.570156 -15.7378 7 13 12 0.86 0.56 - yes Open
2460 8.997477115010753 -0.46383 -13.2881 6 12 0 0.00 0.00 - yes Open
2059 9.123046795785138 -0.794823 -18.14 9 17 0 0.00 0.00 - yes Open
2061 9.741765202331994 -0.676692 -19.0511 8 18 0 0.00 0.00 - yes Open
2458 10.051436411354386 -0.589233 -12.4988 5 10 0 0.00 0.00 - yes Open
2066 12.229632591397024 -0.717067 -22.6047 7 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.793kcal/mol
Ligand efficiency (LE) -0.5417kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.278
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 418.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.87
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.09kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 104.72kcal/mol
Minimised FF energy 85.63kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.