FAIRMol

OSA_Lib_277

Pose ID 5123 Compound 102 Pose 1805

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.673 kcal/mol/HA) ✓ Good fit quality (FQ -6.74) ✗ Very high strain energy (45.8 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.886
kcal/mol
LE
-0.673
kcal/mol/HA
Fit Quality
-6.74
FQ (Leeson)
HAC
34
heavy atoms
MW
464
Da
LogP
0.41
cLogP
Strain ΔE
45.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 45.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 7 Severe clashes 1
Final rank55.33280609114375Score-22.8862
Inter norm-0.725146Intra norm0.052024
Top1000noExcludedyes
Contacts18H-bonds1
Artifact reasonexcluded; geometry warning; 12 clashes; 1 protein clash
ResiduesA:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER86;A:THR83;A:TRP47;A:VAL156;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.58RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1800 3.192995042814929 -0.666482 -19.5956 1 16 12 0.60 0.00 - no Open
1712 3.852309507173588 -0.740658 -23.1814 1 21 0 0.00 0.00 - no Open
1720 4.041475288126007 -0.711065 -24.1449 1 16 0 0.00 0.00 - no Open
1716 4.39232578635824 -0.682733 -21.5601 1 18 0 0.00 0.00 - no Open
1797 4.573080037112168 -0.732454 -23.9797 1 20 15 0.75 0.20 - no Open
1799 4.576968853356978 -0.701699 -21.5859 1 16 12 0.60 0.20 - no Open
1723 4.645652209172564 -0.740475 -26.1491 1 17 0 0.00 0.00 - no Open
1724 5.324635239472977 -0.715558 -21.0734 1 17 0 0.00 0.00 - no Open
1715 5.329875143919994 -0.657376 -22.1009 0 19 0 0.00 0.00 - no Open
1809 5.7094446096767095 -0.700127 -19.268 1 20 17 0.85 0.20 - no Open
1811 5.7401879531940585 -0.762086 -24.3652 2 18 14 0.70 0.20 - no Open
1721 53.883265066727375 -0.64254 -20.7416 1 15 0 0.00 0.00 - no Open
1722 54.18895745625761 -0.674571 -20.5181 1 18 0 0.00 0.00 - no Open
1714 54.49632132726808 -0.640732 -18.8551 1 17 0 0.00 0.00 - no Open
1719 54.57943991446807 -0.658254 -23.9656 1 18 0 0.00 0.00 - no Open
1802 55.009085085725 -0.789943 -23.4261 1 17 13 0.65 0.20 - no Open
1804 55.3547913067628 -0.716942 -22.6573 1 17 15 0.75 0.00 - no Open
1798 55.57448442123359 -0.716794 -16.8477 1 17 15 0.75 0.20 - no Open
1808 5.258365990403331 -0.691236 -19.0268 2 17 13 0.65 0.00 - yes Open
1807 54.22172094920189 -0.652744 -22.6324 1 17 13 0.65 0.00 - yes Open
1801 54.766080237386284 -0.714425 -23.1078 1 17 13 0.65 0.20 - yes Open
1806 55.01311487972341 -0.676746 -21.1357 2 17 13 0.65 0.00 - yes Open
1713 55.21619935175384 -0.708345 -22.1161 1 19 0 0.00 0.00 - yes Open
1711 55.278694716865154 -0.622768 -18.9073 1 19 0 0.00 0.00 - yes Open
1805 55.33280609114375 -0.725146 -22.8862 1 18 14 0.70 0.20 - yes Current
1812 55.67171030508722 -0.662607 -19.9533 1 18 15 0.75 0.00 - yes Open
1803 55.89989271176973 -0.743185 -25.5761 3 18 16 0.80 0.20 - yes Open
1718 56.34810804689525 -0.579787 -17.7791 0 18 0 0.00 0.00 - yes Open
1710 56.63998815049071 -0.672228 -17.5114 1 18 0 0.00 0.00 - yes Open
1717 56.79149628766385 -0.785071 -23.3202 1 21 0 0.00 0.00 - yes Open
1709 56.973941864856805 -0.662562 -21.0627 1 21 0 0.00 0.00 - yes Open
1810 58.535454443647325 -0.839785 -26.5027 1 20 16 0.80 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.886kcal/mol
Ligand efficiency (LE) -0.6731kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.735
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 463.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.41
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 45.78kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 295.71kcal/mol
Minimised FF energy 249.93kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.