FAIRMol

OSA_Lib_247

Pose ID 5081 Compound 682 Pose 1763

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.616 kcal/mol/HA) ✓ Good fit quality (FQ -6.30) ✗ Very high strain energy (34.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.786
kcal/mol
LE
-0.616
kcal/mol/HA
Fit Quality
-6.30
FQ (Leeson)
HAC
37
heavy atoms
MW
502
Da
LogP
3.22
cLogP
Strain ΔE
34.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 34.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 11 Severe clashes 0
Final rank7.180705676477455Score-22.7859
Inter norm-0.61571Intra norm-0.000126263
Top1000noExcludedno
Contacts17H-bonds1
Artifact reasongeometry warning; 18 clashes; 11 protein contact clashes; high strain Δ 28.3
ResiduesA:ALA32;A:ASP52;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR83;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.76RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1764 6.003681738816833 -0.691597 -23.7488 2 17 16 0.80 0.20 - no Open
2271 6.2343531801697285 -0.521155 -16.39 0 16 0 0.00 0.00 - no Open
2270 6.964934773791494 -0.56824 -15.642 0 17 0 0.00 0.00 - no Open
1763 7.180705676477455 -0.61571 -22.7859 1 17 16 0.80 0.00 - no Current
1761 6.860347609611279 -0.671427 -22.8152 0 21 16 0.80 0.00 - yes Open
2269 7.029889752638729 -0.629109 -22.114 2 17 0 0.00 0.00 - yes Open
1762 57.015733488828715 -0.620626 -18.1674 0 16 14 0.70 0.00 - yes Open
2268 57.15484765343514 -0.554568 -19.3039 2 13 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.786kcal/mol
Ligand efficiency (LE) -0.6158kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.305
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 501.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.22
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 33.99kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 104.06kcal/mol
Minimised FF energy 70.07kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.