FAIRMol

OSA_Lib_78

Pose ID 50526 Compound 3555 Pose 670

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.588 kcal/mol/HA) ✓ Good fit quality (FQ -6.02) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (32.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.771
kcal/mol
LE
-0.588
kcal/mol/HA
Fit Quality
-6.02
FQ (Leeson)
HAC
37
heavy atoms
MW
504
Da
LogP
3.54
cLogP
Strain ΔE
32.9 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 8 π–π 1 Clashes 7 Severe clashes 0
Final rank6.557381766036804Score-21.7709
Inter norm-0.593662Intra norm0.00525924
Top1000noExcludedno
Contacts17H-bonds5
Artifact reasongeometry warning; 18 clashes; 7 protein contact clashes; high strain Δ 32.0
ResiduesA:ARG137;A:ARG141;A:ASN103;A:HIS102;A:MET98;A:TYR94;B:ARG113;B:ASP10;B:CYS69;B:GLY70;B:GLY72;B:GLY74;B:HIS11;B:ILE73;B:PRO12;B:SER71;B:TYR46

Protein summary

305 residues
Protein targetT21Atoms4646
Residues305Chains2
Residue summaryARG:576; ILE:532; VAL:512; GLU:420; ALA:360; PHE:240; HIS:238; LYS:220; THR:210; LEU:190; PRO:168; TYR:168; GLY:154; SER:154; ASP:144; ASN:112

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3K7OContacts14
PoseOpen native poseH-bonds16
IFP residuesA:ARG137; A:ARG141; A:ASN103; A:HIS102; A:HIS138; B:ASP10; B:CYS69; B:GLY70; B:GLY74; B:HIS11; B:ILE73; B:PRO12; B:SER71; B:TYR46
Current overlap13Native recall0.93
Jaccard0.72RMSD-
H-bond strict4Strict recall0.33
H-bond same residue+role4Role recall0.44
H-bond same residue4Residue recall0.50

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
654 5.214036576432896 -0.68265 -25.2249 6 16 13 0.93 0.44 - no Open
673 5.7077034443090096 -0.616642 -24.8958 6 13 13 0.93 0.56 - no Open
658 5.9237349254497556 -0.593119 -21.5278 6 18 14 1.00 0.44 - no Open
657 6.235073014560082 -0.615329 -22.2864 5 15 13 0.93 0.44 - no Open
670 6.557381766036804 -0.593662 -21.7709 5 17 13 0.93 0.44 - no Current
672 7.490409203869804 -0.570146 -8.92039 4 15 13 0.93 0.33 - no Open
664 55.73728239861711 -0.517254 -20.6854 6 14 12 0.86 0.22 - no Open
662 56.231200613246614 -0.51026 -15.1571 4 16 13 0.93 0.22 - no Open
667 56.303877576902465 -0.418416 -13.8344 5 13 11 0.79 0.22 - no Open
660 55.60911231374396 -0.518593 -16.0694 5 15 13 0.93 0.44 - yes Open
656 55.62076309807943 -0.688986 -21.0343 5 17 13 0.93 0.33 - yes Open
668 55.84970052370133 -0.629089 -20.306 4 16 13 0.93 0.33 - yes Open
674 56.165025313900884 -0.587024 -21.5238 6 18 14 1.00 0.44 - yes Open
653 56.57847877966354 -0.554913 -15.9633 9 17 13 0.93 0.56 - yes Open
652 56.64543113536261 -0.510289 -20.1753 2 15 12 0.86 0.22 - yes Open
655 56.6668739453166 -0.665607 -22.5798 6 15 12 0.86 0.44 - yes Open
663 56.763290574356795 -0.574524 -19.7033 4 16 13 0.93 0.33 - yes Open
665 56.889727510317954 -0.436431 -16.5985 4 15 13 0.93 0.33 - yes Open
671 57.0134770838262 -0.608412 -19.8882 2 15 12 0.86 0.22 - yes Open
669 57.209848642128776 -0.492448 -18.2303 6 16 13 0.93 0.44 - yes Open
651 57.46282018486445 -0.66688 -21.2643 5 18 14 1.00 0.44 - yes Open
661 58.01173561173015 -0.528289 -13.0474 7 14 11 0.79 0.44 - yes Open
659 58.05077495714546 -0.483489 -14.0542 5 14 11 0.79 0.33 - yes Open
666 61.76193635208182 -0.496801 -10.9901 6 14 12 0.86 0.33 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.771kcal/mol
Ligand efficiency (LE) -0.5884kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.024
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 503.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.54
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 32.85kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 109.57kcal/mol
Minimised FF energy 76.72kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.