FAIRMol

OSA_Lib_239

Pose ID 5005 Compound 529 Pose 1687

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.818 kcal/mol/HA) ✓ Good fit quality (FQ -7.89) ✗ Very high strain energy (41.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-24.545
kcal/mol
LE
-0.818
kcal/mol/HA
Fit Quality
-7.89
FQ (Leeson)
HAC
30
heavy atoms
MW
406
Da
LogP
1.85
cLogP
Strain ΔE
41.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 41.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 8 Severe clashes 0
Final rank54.68616997773502Score-24.5454
Inter norm-0.844469Intra norm0.0262902
Top1000noExcludedno
Contacts20H-bonds1
Artifact reasongeometry warning; 14 clashes; 8 protein contact clashes
ResiduesA:ALA32;A:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PRO88;A:SER86;A:THR54;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.74RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1679 3.8211097807997416 -0.858111 -25.7538 0 21 18 0.90 0.00 - no Open
1682 3.84020984989632 -0.710977 -20.9194 0 16 16 0.80 0.00 - no Open
1674 3.934725849205876 -0.721152 -21.6615 0 18 15 0.75 0.00 - no Open
1681 4.300761839522966 -0.688906 -20.3079 0 19 15 0.75 0.00 - no Open
1678 4.337918151361544 -0.681481 -18.9776 0 18 15 0.75 0.00 - no Open
1683 4.410761028776333 -0.647598 -20.1427 0 18 15 0.75 0.00 - no Open
1688 53.53925770848332 -0.702991 -18.1506 2 19 16 0.80 0.20 - no Open
1673 53.59461909940166 -0.631063 -16.4089 0 17 17 0.85 0.00 - no Open
1680 54.250888920292375 -0.703922 -19.1243 1 18 17 0.85 0.00 - no Open
1675 54.557920964248666 -0.664692 -19.5125 0 18 14 0.70 0.00 - no Open
1687 54.68616997773502 -0.844469 -24.5454 1 20 17 0.85 0.00 - no Current
1676 54.87589185365573 -0.68266 -19.8441 0 15 11 0.55 0.00 - no Open
1684 54.9344767219574 -0.699194 -21.0605 0 16 12 0.60 0.00 - no Open
1685 55.24792418956906 -0.719354 -17.7936 1 19 16 0.80 0.20 - no Open
1686 55.796250310983375 -0.81184 -20.8051 1 18 15 0.75 0.20 - no Open
1677 54.90345637625511 -0.726472 -19.0427 0 18 15 0.75 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.545kcal/mol
Ligand efficiency (LE) -0.8182kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.892
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 405.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.85
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 40.98kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 106.72kcal/mol
Minimised FF energy 65.74kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.