FAIRMol

OSA_Lib_237

Pose ID 4981 Compound 581 Pose 1663

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.690 kcal/mol/HA) ✓ Good fit quality (FQ -6.85) ✗ Very high strain energy (22.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.770
kcal/mol
LE
-0.690
kcal/mol/HA
Fit Quality
-6.85
FQ (Leeson)
HAC
33
heavy atoms
MW
446
Da
LogP
2.77
cLogP
Strain ΔE
22.8 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 22.8 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 8 Severe clashes 0
Final rank54.95178217854325Score-22.7696
Inter norm-0.70715Intra norm0.0171621
Top1000noExcludedno
Contacts17H-bonds1
Artifact reasongeometry warning; 15 clashes; 8 protein contact clashes
ResiduesA:ALA32;A:ARG48;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:THR83;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.61RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1216 4.013882301094123 -0.502014 -17.8447 3 11 0 0.00 0.00 - no Open
1212 4.396990726588747 -0.454885 -15.7572 2 10 0 0.00 0.00 - no Open
1664 4.642272634384539 -0.786068 -23.9847 1 19 18 0.90 0.20 - no Open
1213 4.82058525967209 -0.519629 -17.2292 3 11 0 0.00 0.00 - no Open
1660 5.053914738507422 -0.65804 -23.2919 1 18 17 0.85 0.20 - no Open
1662 5.609317620858329 -0.694604 -24.6632 1 21 17 0.85 0.00 - no Open
1215 54.014337055346104 -0.565989 -17.3348 2 9 0 0.00 0.00 - no Open
1211 54.49758931621311 -0.545004 -15.1878 3 9 0 0.00 0.00 - no Open
1658 54.67424900407422 -0.722052 -24.1029 1 12 9 0.45 0.20 - no Open
1663 54.95178217854325 -0.70715 -22.7696 1 17 14 0.70 0.00 - no Current
1210 55.012375243918925 -0.493339 -18.3483 4 11 0 0.00 0.00 - no Open
1214 55.050565107588966 -0.502724 -18.594 3 10 0 0.00 0.00 - no Open
1661 55.52037280295748 -0.780499 -26.2914 1 18 15 0.75 0.20 - no Open
1209 54.94606519573975 -0.359535 -13.2979 1 11 0 0.00 0.00 - yes Open
1657 56.02607467946437 -0.705187 -20.9165 0 18 15 0.75 0.00 - yes Open
1659 58.524733583480845 -0.729517 -24.9158 1 19 16 0.80 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.770kcal/mol
Ligand efficiency (LE) -0.6900kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.846
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 445.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.77
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.82kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 93.42kcal/mol
Minimised FF energy 70.60kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.