FAIRMol

Z56175983

Pose ID 49808 Compound 3290 Pose 2843

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.463 kcal/mol/HA) ✓ Good fit quality (FQ -4.42) ✓ Strong H-bond network (7 bonds) ✗ Very high strain energy (39.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-13.426
kcal/mol
LE
-0.463
kcal/mol/HA
Fit Quality
-4.42
FQ (Leeson)
HAC
29
heavy atoms
MW
387
Da
LogP
4.55
cLogP
Strain ΔE
39.2 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 7 Hydrophobic 13 π–π 1 Clashes 8 Severe clashes 0
Final rank8.050501809021219Score-13.4264
Inter norm-0.606442Intra norm0.143462
Top1000noExcludedno
Contacts6H-bonds7
Artifact reasongeometry warning; 17 clashes; 8 protein contact clashes; high strain Δ 55.9
ResiduesA:ASN402;A:LEU399;A:LYS407;A:PHE396;A:PRO398;A:THR397

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap5Native recall0.62
Jaccard0.56RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2187 6.72959580888413 -1.10709 -27.8499 5 20 0 0.00 0.00 - no Open
2844 6.802451193186113 -0.661541 -16.926 5 7 6 0.75 0.00 - no Open
2843 8.050501809021219 -0.606442 -13.4264 7 6 5 0.62 0.00 - no Current
2189 8.185745733851823 -1.21552 -33.1116 6 17 0 0.00 0.00 - no Open
2845 7.783379389481876 -0.565641 -15.82 7 7 6 0.75 0.00 - yes Open
2191 9.954485767120143 -1.11811 -30.5533 6 18 0 0.00 0.00 - yes Open
2188 10.082435984622862 -1.0252 -28.9828 5 19 0 0.00 0.00 - yes Open
2846 10.44678636690243 -0.604876 -17.3176 7 8 7 0.88 0.00 - yes Open
2190 11.565762983648456 -1.06908 -30.7692 4 22 0 0.00 0.00 - yes Open
2186 12.399546710458454 -1.06826 -29.767 8 21 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -13.426kcal/mol
Ligand efficiency (LE) -0.4630kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.419
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 29HA

Physicochemical properties

Molecular weight 387.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.55
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.16kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 91.14kcal/mol
Minimised FF energy 51.97kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.