FAIRMol

Z49620424

Pose ID 49387 Compound 3112 Pose 2422

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.853 kcal/mol/HA) ✓ Good fit quality (FQ -7.86) ✓ Good H-bonds (5 bonds) ✗ High strain energy (19.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.184
kcal/mol
LE
-0.853
kcal/mol/HA
Fit Quality
-7.86
FQ (Leeson)
HAC
26
heavy atoms
MW
344
Da
LogP
3.80
cLogP
Strain ΔE
19.5 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 16 π–π 3 Clashes 7 Severe clashes 0
Final rank5.083538880826211Score-22.1843
Inter norm-0.648994Intra norm-0.204247
Top1000noExcludedno
Contacts12H-bonds5
Artifact reasongeometry warning; 15 clashes; 7 protein contact clashes; moderate strain Δ 19.9
ResiduesA:ASN402;A:GLU466;A:GLU467;A:HIS461;A:LEU399;A:PHE396;A:PRO398;A:PRO462;A:SER394;A:SER395;A:THR397;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap7Native recall0.88
Jaccard0.54RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2258 4.432800924488171 -0.535128 -19.4395 5 7 0 0.00 0.00 - no Open
2257 4.835953911856199 -0.744747 -19.5352 3 14 0 0.00 0.00 - no Open
2418 4.880178323318226 -0.53481 -16.8962 3 10 8 1.00 0.00 - no Open
2422 5.083538880826211 -0.648994 -22.1843 5 12 7 0.88 0.00 - no Current
2414 5.111839317552878 -0.724754 -21.3757 5 12 7 0.88 0.00 - no Open
2262 5.269524950228686 -0.519459 -17.7185 2 11 0 0.00 0.00 - no Open
2420 5.484780132869905 -0.583976 -18.8854 4 11 7 0.88 0.00 - no Open
2263 5.700764560190182 -0.585764 -12.6616 3 9 0 0.00 0.00 - no Open
2423 5.977953095303983 -0.51653 -10.2878 4 9 6 0.75 0.00 - no Open
2416 5.521791695792289 -0.621012 -21.9887 4 8 7 0.88 0.00 - yes Open
2419 5.594801201247525 -0.590564 -13.9392 3 13 8 1.00 0.00 - yes Open
2261 5.62039704457523 -0.797512 -19.6201 3 14 0 0.00 0.00 - yes Open
2415 6.120347422726654 -0.674279 -15.7188 3 13 8 1.00 0.00 - yes Open
2424 6.7205022423280765 -0.725098 -24.6134 5 11 7 0.88 0.00 - yes Open
2255 7.208832376833763 -0.633863 -12.6031 5 14 0 0.00 0.00 - yes Open
2259 7.5292507820024985 -0.549638 -12.3161 6 14 0 0.00 0.00 - yes Open
2264 8.646106306293484 -0.609641 -19.9337 6 15 0 0.00 0.00 - yes Open
2256 9.651344200099961 -0.852122 -18.7429 5 14 0 0.00 0.00 - yes Open
2417 56.04513878602127 -0.717115 -23.5487 5 12 7 0.88 0.00 - yes Open
2421 56.32837484254128 -0.608588 -24.2175 4 12 7 0.88 0.00 - yes Open
2425 56.46456058031302 -0.694483 -24.6973 5 12 7 0.88 0.00 - yes Open
2265 57.1115727236319 -0.664429 -16.337 4 14 0 0.00 0.00 - yes Open
2254 58.505358458890775 -0.549167 -18.9903 5 11 0 0.00 0.00 - yes Open
2260 58.95205146539992 -0.723753 -20.0449 3 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.184kcal/mol
Ligand efficiency (LE) -0.8532kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.861
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 26HA

Physicochemical properties

Molecular weight 344.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.80
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.54kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 105.70kcal/mol
Minimised FF energy 86.16kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.