FAIRMol

Z56891526

Pose ID 49348 Compound 1309 Pose 2383

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.984 kcal/mol/HA) ✓ Good fit quality (FQ -8.06) ✓ Strong H-bond network (6 bonds) ✗ High strain energy (19.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-18.690
kcal/mol
LE
-0.984
kcal/mol/HA
Fit Quality
-8.06
FQ (Leeson)
HAC
19
heavy atoms
MW
280
Da
LogP
-0.53
cLogP
Strain ΔE
19.5 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 6 Hydrophobic 12 π–π 2 Clashes 4 Severe clashes 0
Final rank3.3691070679647694Score-18.6897
Inter norm-0.959669Intra norm-0.0239967
Top1000noExcludedno
Contacts8H-bonds6
Artifact reasongeometry warning; 5 clashes; 4 protein contact clashes; high strain Δ 38.9
ResiduesA:ASN402;A:GLU467;A:LEU399;A:PHE396;A:PRO398;A:SER394;A:SER395;A:THR397

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap7Native recall0.88
Jaccard0.78RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1728 1.8768500769955772 -1.46993 -26.9835 9 11 0 0.00 0.00 - no Open
1745 1.9834483987050242 -1.4796 -24.9362 6 15 0 0.00 0.00 - no Open
1733 2.228029426087275 -1.56417 -24.0185 8 14 0 0.00 0.00 - no Open
1749 2.6686075151339974 -1.40889 -22.7764 7 13 0 0.00 0.00 - no Open
2384 2.7665709012998856 -0.800212 -10.3619 7 10 8 1.00 1.00 - no Open
2386 3.063855139650708 -0.705845 -15.1068 4 11 6 0.75 1.00 - no Open
2383 3.3691070679647694 -0.959669 -18.6897 6 8 7 0.88 0.00 - no Current
2380 3.7728355845938437 -0.868045 -13.6551 4 6 5 0.62 0.00 - no Open
2381 4.192362665201653 -0.926177 -14.9424 5 9 6 0.75 1.00 - no Open
2387 4.027534994665723 -0.774964 -17.7489 3 12 6 0.75 1.00 - yes Open
1730 4.184816189649055 -1.57481 -31.1023 9 13 0 0.00 0.00 - yes Open
2376 4.195270266235503 -0.772547 -11.2454 6 10 8 1.00 1.00 - yes Open
1736 4.235644058595453 -1.72474 -30.9389 12 13 0 0.00 0.00 - yes Open
1740 4.362540520889233 -1.5377 -28.1586 13 14 0 0.00 0.00 - yes Open
2379 4.395695783244731 -0.691419 -14.7706 2 12 6 0.75 1.00 - yes Open
1737 4.471584691160689 -1.48494 -23.8955 13 12 0 0.00 0.00 - yes Open
2375 4.590753002006133 -0.827752 -15.665 6 6 5 0.62 1.00 - yes Open
2374 4.648031556519652 -0.738606 -14.4039 3 9 5 0.62 0.00 - yes Open
1731 4.687035226113764 -1.49332 -29.8656 7 15 0 0.00 0.00 - yes Open
1724 4.733114329638083 -1.81285 -31.3278 13 14 0 0.00 0.00 - yes Open
1725 5.070475388954626 -1.563 -22.8651 9 16 0 0.00 0.00 - yes Open
1748 5.191030239372292 -1.61044 -26.3482 12 13 0 0.00 0.00 - yes Open
1750 5.350947100194247 -1.72325 -31.1372 10 13 0 0.00 0.00 - yes Open
1746 5.422463829297065 -1.53361 -30.1418 10 15 0 0.00 0.00 - yes Open
1732 5.789168079486881 -1.49176 -26.5702 12 12 0 0.00 0.00 - yes Open
1720 5.844183254661189 -1.60197 -27.377 13 14 0 0.00 0.00 - yes Open
2377 5.91533057492604 -0.814325 -14.8362 7 10 6 0.75 1.00 - yes Open
2373 5.964246747470154 -0.932802 -14.2765 5 8 5 0.62 0.00 - yes Open
1743 6.017278855873055 -1.5126 -30.6945 10 14 0 0.00 0.00 - yes Open
1727 6.0228273266289385 -1.77901 -33.9013 11 14 0 0.00 0.00 - yes Open
1735 6.047166506282892 -1.60349 -31.8335 10 14 0 0.00 0.00 - yes Open
1747 6.090022499357254 -1.46347 -31.2729 10 15 0 0.00 0.00 - yes Open
1723 6.2173732351415385 -1.76481 -33.8778 10 15 0 0.00 0.00 - yes Open
1739 6.432889719420583 -1.49872 -28.1324 10 14 0 0.00 0.00 - yes Open
1721 6.6873148479210744 -1.68278 -27.1559 11 14 0 0.00 0.00 - yes Open
1742 6.870627313515039 -1.65378 -31.4661 11 14 0 0.00 0.00 - yes Open
1729 53.68157246368138 -1.55262 -25.3144 10 15 0 0.00 0.00 - yes Open
2385 54.4463891797473 -0.779176 -13.8316 6 10 6 0.75 1.00 - yes Open
2382 54.64345394835052 -0.607939 -8.72254 5 5 5 0.62 0.00 - yes Open
1751 54.67885502729105 -1.62829 -31.6119 10 13 0 0.00 0.00 - yes Open
2372 55.102080780144014 -0.881783 -13.7554 5 10 6 0.75 0.00 - yes Open
1738 55.28656080891448 -1.76052 -31.9977 12 14 0 0.00 0.00 - yes Open
2378 55.46882946601546 -0.722593 -14.837 5 6 5 0.62 0.00 - yes Open
1744 55.81541597793679 -1.40235 -26.5901 5 14 0 0.00 0.00 - yes Open
1741 56.14817845781458 -1.33485 -19.8743 9 16 0 0.00 0.00 - yes Open
1726 56.26815783120112 -1.94463 -34.8227 13 14 0 0.00 0.00 - yes Open
1734 56.43104277264373 -1.67285 -30.1159 11 12 0 0.00 0.00 - yes Open
1722 56.46358177993412 -1.77833 -31.4787 11 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.690kcal/mol
Ligand efficiency (LE) -0.9837kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.063
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 19HA

Physicochemical properties

Molecular weight 280.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.53
Lipinski: ≤ 5
Rotatable bonds 2

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.50kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 90.95kcal/mol
Minimised FF energy 71.46kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.