FAIRMol

OSA_Lib_228

Pose ID 4921 Compound 485 Pose 1603

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.535 kcal/mol/HA) ✓ Good fit quality (FQ -5.35) ✗ Very high strain energy (30.2 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-18.188
kcal/mol
LE
-0.535
kcal/mol/HA
Fit Quality
-5.35
FQ (Leeson)
HAC
34
heavy atoms
MW
464
Da
LogP
0.11
cLogP
Strain ΔE
30.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 30.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 10 Severe clashes 1
Final rank56.784558556448395Score-18.1878
Inter norm-0.629064Intra norm0.0941281
Top1000noExcludedyes
Contacts18H-bonds2
Artifact reasonexcluded; geometry warning; 14 clashes; 1 protein clash
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR180;A:TRP47;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.58RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1605 3.1588074003271673 -0.608688 -18.5717 0 17 13 0.65 0.00 - no Open
1618 3.8369003827623267 -0.64116 -20.2576 1 18 14 0.70 0.00 - no Open
1601 3.93144186678271 -0.715903 -22.8001 0 17 14 0.70 0.00 - no Open
1602 4.320292172863569 -0.732107 -20.8356 0 18 14 0.70 0.00 - no Open
1613 4.678370170206609 -0.691038 -22.6808 2 19 14 0.70 0.20 - no Open
1615 4.8022510309289475 -0.591258 -13.641 1 17 16 0.80 0.20 - no Open
1616 5.216230902400127 -0.694483 -22.2258 2 19 15 0.75 0.00 - no Open
1620 5.344845183894786 -0.636657 -17.143 0 18 14 0.70 0.00 - no Open
1617 5.683183286281492 -0.798681 -23.9269 1 19 15 0.75 0.20 - no Open
1606 53.31267611278559 -0.667379 -21.6326 1 16 12 0.60 0.00 - no Open
1608 53.316965812699 -0.649911 -21.2635 2 18 15 0.75 0.20 - no Open
1604 53.538090361062245 -0.786872 -27.1379 1 19 16 0.80 0.00 - no Open
1609 54.08163966417761 -0.728123 -20.9196 1 18 15 0.75 0.00 - no Open
1610 55.086836897863975 -0.797384 -25.6545 1 18 14 0.70 0.20 - no Open
1614 55.35975567749378 -0.675678 -22.5696 2 19 14 0.70 0.20 - yes Open
1612 55.668143165071875 -0.812916 -22.9737 1 19 15 0.75 0.20 - yes Open
1611 56.28313283384909 -0.697023 -24.4572 1 17 16 0.80 0.00 - yes Open
1619 56.502378095906494 -0.721697 -19.705 0 19 15 0.75 0.00 - yes Open
1603 56.784558556448395 -0.629064 -18.1878 2 18 14 0.70 0.20 - yes Current
1607 56.87477982360974 -0.66658 -18.8594 0 18 15 0.75 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.188kcal/mol
Ligand efficiency (LE) -0.5349kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.353
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 463.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.11
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 30.23kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 282.59kcal/mol
Minimised FF energy 252.36kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.