FAIRMol

Z29884022

Pose ID 48986 Compound 3305 Pose 2021

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.630 kcal/mol/HA) ✓ Good fit quality (FQ -5.73) ✓ Good H-bonds (3 bonds) ✗ Moderate strain (8.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-15.760
kcal/mol
LE
-0.630
kcal/mol/HA
Fit Quality
-5.73
FQ (Leeson)
HAC
25
heavy atoms
MW
337
Da
LogP
3.24
cLogP
Strain ΔE
8.0 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 13 π–π 1 Clashes 4 Severe clashes 0 ⚠ Hydrophobic exposure 50%
⚠️Partial hydrophobic solvent exposure
50% of hydrophobic surface appears solvent-exposed (10/20 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 20 Buried (contacted) 10 Exposed 10 LogP 3.24 H-bonds 3
Exposed fragments: phenyl (4/6 atoms exposed)phenyl (6/6 atoms exposed)aliphatic chain/group (2 atoms exposed)
Final rank2.59361117049877Score-15.7602
Inter norm-0.642644Intra norm0.0122377
Top1000noExcludedno
Contacts9H-bonds3
Artifact reasongeometry warning; 8 clashes; 4 protein contact clashes; moderate strain Δ 12.5
ResiduesA:ASN402;A:GLU467;A:LEU399;A:LYS407;A:LYS410;A:PHE396;A:PRO398;A:SER394;A:THR397

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap7Native recall0.88
Jaccard0.70RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2021 2.59361117049877 -0.642644 -15.7602 3 9 7 0.88 0.00 - no Current
2020 6.1547261910267785 -0.765945 -14.7722 3 9 6 0.75 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -15.760kcal/mol
Ligand efficiency (LE) -0.6304kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.731
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 337.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.24
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 8.04kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 67.51kcal/mol
Minimised FF energy 59.47kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.