FAIRMol

Z30225126

Pose ID 48854 Compound 1880 Pose 1889

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.531 kcal/mol/HA) ✓ Good fit quality (FQ -5.17) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (22.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-16.461
kcal/mol
LE
-0.531
kcal/mol/HA
Fit Quality
-5.17
FQ (Leeson)
HAC
31
heavy atoms
MW
460
Da
LogP
3.18
cLogP
Strain ΔE
22.3 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 5 π–π 1 Clashes 7 Severe clashes 0
Final rank4.694512282184984Score-16.4608
Inter norm-0.468798Intra norm-0.0621948
Top1000noExcludedno
Contacts11H-bonds4
Artifact reasongeometry warning; 11 clashes; 7 protein contact clashes; high strain Δ 21.9
ResiduesA:GLU466;A:GLU467;A:HIS461;A:MET393;A:MET471;A:PHE396;A:PRO462;A:SER394;A:SER395;A:SER470;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap4Native recall0.50
Jaccard0.27RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1539 4.239954776220724 -0.800001 -24.6016 2 19 0 0.00 0.00 - no Open
1538 4.486289734677165 -0.809436 -24.9924 2 16 0 0.00 0.00 - no Open
1889 4.694512282184984 -0.468798 -16.4608 4 11 4 0.50 1.00 - no Current
1888 8.434483896025103 -0.585574 -18.194 4 12 8 1.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.461kcal/mol
Ligand efficiency (LE) -0.5310kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.173
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 459.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.18
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.27kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -37.29kcal/mol
Minimised FF energy -59.56kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.