FAIRMol

OHD_MAC_16

Pose ID 48697 Compound 1015 Pose 1732

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good fit quality (FQ -1.81) ✓ Strong H-bond network (8 bonds) ✗ Very high strain energy (22.2 kcal/mol) ✗ Low LE (-0.183 kcal/mol/HA) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-6.024
kcal/mol
LE
-0.183
kcal/mol/HA
Fit Quality
-1.81
FQ (Leeson)
HAC
33
heavy atoms
MW
447
Da
LogP
2.78
cLogP
Strain ΔE
22.2 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 8 Hydrophobic 12 π–π 1 Clashes 8 Severe clashes 0 ⚠ Hydrophobic exposure 45%
⚠️Partial hydrophobic solvent exposure
45% of hydrophobic surface appears solvent-exposed (10/22 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 22 Buried (contacted) 12 Exposed 10 LogP 2.78 H-bonds 8
Exposed fragments: phenyl (6/6 atoms exposed)aliphatic chain/group (4 atoms exposed)
Final rank6.658729660090414Score-6.02426
Inter norm-0.440653Intra norm0.2581
Top1000noExcludedno
Contacts9H-bonds8
Artifact reasongeometry warning; 15 clashes; 8 protein contact clashes; high strain Δ 35.1
ResiduesA:ASN402;A:GLU467;A:LEU399;A:LYS407;A:PHE396;A:PRO398;A:SER470;A:THR397;A:TYR455

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap7Native recall0.88
Jaccard0.70RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1299 5.752180216571295 -0.768978 -16.8738 3 19 0 0.00 0.00 - no Open
827 6.406292800265652 -0.596367 -11.4458 5 13 0 0.00 0.00 - no Open
1303 6.465793938784395 -0.635253 -15.7051 2 18 0 0.00 0.00 - no Open
1050 6.54588703754338 -0.984045 -28.9382 8 21 0 0.00 0.00 - no Open
1732 6.658729660090414 -0.440653 -6.02426 8 9 7 0.88 1.00 - no Current
3130 7.382563025709787 -0.550936 -9.26817 3 15 0 0.00 0.00 - no Open
1049 7.568665222351072 -0.964885 -23.2533 12 18 0 0.00 0.00 - no Open
795 9.144947144102693 -0.689423 -14.8045 7 16 0 0.00 0.00 - no Open
831 6.477716366125133 -0.65885 -13.2458 3 16 0 0.00 0.00 - yes Open
1729 6.892186765656801 -0.472582 -10.4809 7 12 8 1.00 1.00 - yes Open
830 6.921351728111539 -0.614096 -10.0328 5 13 0 0.00 0.00 - yes Open
3131 7.715012804359663 -0.542545 -14.4034 4 13 0 0.00 0.00 - yes Open
1733 7.779429151432847 -0.492017 -9.69993 7 10 7 0.88 1.00 - yes Open
1054 7.7850298411484715 -0.884636 -25.6916 8 19 0 0.00 0.00 - yes Open
1053 7.910783283220195 -0.921235 -24.2883 11 19 0 0.00 0.00 - yes Open
796 8.275569663309865 -0.684241 -18.6059 9 15 0 0.00 0.00 - yes Open
1734 8.465194828859476 -0.489927 -11.5371 9 11 8 1.00 1.00 - yes Open
1056 8.53325070554073 -0.919496 -24.7526 9 16 0 0.00 0.00 - yes Open
791 8.755780369521949 -0.763071 -14.473 15 9 0 0.00 0.00 - yes Open
1730 8.918006274137584 -0.583552 -16.8151 7 17 8 1.00 0.00 - yes Open
1055 9.346918705545136 -0.879942 -25.302 8 16 0 0.00 0.00 - yes Open
1302 9.3534034729308 -0.615452 -10.8719 5 19 0 0.00 0.00 - yes Open
832 9.441916496247993 -0.632948 -16.0685 9 12 0 0.00 0.00 - yes Open
829 9.451566458846896 -0.677978 -6.62565 3 15 0 0.00 0.00 - yes Open
3126 9.50785916439563 -0.694616 -16.7147 6 20 0 0.00 0.00 - yes Open
1304 9.764372204867888 -0.72286 -19.2905 3 13 0 0.00 0.00 - yes Open
1301 10.310890285662667 -0.851027 -14.1153 5 18 0 0.00 0.00 - yes Open
3132 10.444857375642064 -0.778666 -16.8779 4 17 0 0.00 0.00 - yes Open
3127 10.531440804148529 -0.780129 -20.4372 5 17 0 0.00 0.00 - yes Open
3128 10.599414779357968 -0.657745 -16.0162 3 15 0 0.00 0.00 - yes Open
3129 10.850975383060266 -0.552587 -12.4876 4 15 0 0.00 0.00 - yes Open
792 10.853850896897907 -0.786848 -20.8854 12 11 0 0.00 0.00 - yes Open
828 11.056936513202471 -0.670967 -15.8784 8 16 0 0.00 0.00 - yes Open
1300 11.184958117667579 -0.84987 -23.53 5 18 0 0.00 0.00 - yes Open
1731 12.034641062842804 -0.434355 -8.65102 7 11 7 0.88 0.00 - yes Open
793 12.18267700845879 -0.785489 -11.3927 16 14 0 0.00 0.00 - yes Open
794 12.285590442450683 -0.930086 -25.1977 9 23 0 0.00 0.00 - yes Open
1052 13.376173420751345 -1.28243 -31.5208 10 17 0 0.00 0.00 - yes Open
1051 13.39531970759979 -1.1525 -28.5081 8 17 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -6.024kcal/mol
Ligand efficiency (LE) -0.1826kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -1.811
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 447.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.78
Lipinski: ≤ 5
Rotatable bonds 9

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.22kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 86.17kcal/mol
Minimised FF energy 63.95kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.