FAIRMol

OSA_Lib_313

Pose ID 48256 Compound 3394 Pose 1291

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.478 kcal/mol/HA) ✓ Good fit quality (FQ -5.08) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (35.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.556
kcal/mol
LE
-0.478
kcal/mol/HA
Fit Quality
-5.08
FQ (Leeson)
HAC
43
heavy atoms
MW
580
Da
LogP
5.20
cLogP
Strain ΔE
35.5 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 21 π–π 2 Clashes 3 Severe clashes 0
Final rank5.317353963996452Score-20.5557
Inter norm-0.487617Intra norm0.00957824
Top1000noExcludedno
Contacts14H-bonds3
Artifact reasongeometry warning; 17 clashes; 3 protein contact clashes; high strain Δ 34.6
ResiduesA:ASN402;A:GLU466;A:GLU467;A:HIS461;A:LEU399;A:LYS407;A:PHE396;A:PRO398;A:PRO462;A:SER394;A:SER464;A:SER470;A:THR397;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap8Native recall1.00
Jaccard0.57RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1291 5.317353963996452 -0.487617 -20.5557 3 14 8 1.00 0.00 - no Current
1290 6.854823735699815 -0.340061 -14.3389 1 11 8 1.00 0.00 - no Open
1289 8.291950524649575 -0.33272 -15.0187 0 12 7 0.88 0.00 - yes Open
1292 58.02144262378672 -0.369256 -13.8098 3 12 8 1.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.556kcal/mol
Ligand efficiency (LE) -0.4780kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.080
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 43HA

Physicochemical properties

Molecular weight 579.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.20
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 35.52kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 138.63kcal/mol
Minimised FF energy 103.11kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.