FAIRMol

OSA_Lib_235

Pose ID 48160 Compound 3318 Pose 1195

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.427 kcal/mol/HA) ✓ Good fit quality (FQ -4.23) ✗ Very high strain energy (27.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-14.077
kcal/mol
LE
-0.427
kcal/mol/HA
Fit Quality
-4.23
FQ (Leeson)
HAC
33
heavy atoms
MW
447
Da
LogP
1.40
cLogP
Strain ΔE
27.0 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 16 π–π 1 Clashes 5 Severe clashes 0
Final rank53.79835748410926Score-14.0772
Inter norm-0.44713Intra norm0.0205466
Top1000noExcludedno
Contacts10H-bonds2
Artifact reasongeometry warning; 12 clashes; 5 protein contact clashes
ResiduesA:ASN402;A:GLU467;A:LEU399;A:MET400;A:PHE396;A:PRO398;A:SER394;A:SER464;A:THR397;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap7Native recall0.88
Jaccard0.64RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1185 3.218718001403164 -0.438748 -12.0836 3 11 5 0.62 1.00 - no Open
1194 3.311023962496338 -0.542937 -14.613 4 13 7 0.88 1.00 - no Open
1196 3.3458521595805992 -0.457294 -12.9177 2 9 7 0.88 0.00 - no Open
1186 3.654785467957428 -0.548217 -16.2995 3 13 7 0.88 1.00 - no Open
1199 4.314934661400124 -0.512084 -12.4789 3 11 7 0.88 1.00 - no Open
1189 4.666449288760196 -0.447328 -13.2361 2 11 6 0.75 1.00 - no Open
1193 53.205469042306454 -0.480592 -9.55289 3 12 6 0.75 1.00 - no Open
1197 53.27280869115642 -0.497584 -13.8393 2 12 7 0.88 0.00 - no Open
1200 53.426897307710774 -0.436809 -10.9747 3 13 6 0.75 1.00 - no Open
1192 53.64971069060668 -0.413963 -12.241 2 13 8 1.00 0.00 - no Open
1198 53.775909854403665 -0.539379 -15.9604 2 10 7 0.88 0.00 - no Open
1195 53.79835748410926 -0.44713 -14.0772 2 10 7 0.88 0.00 - no Current
1188 54.66362997207979 -0.476214 -15.243 2 13 7 0.88 1.00 - no Open
1191 54.10908608581006 -0.475324 -14.6419 2 11 7 0.88 0.00 - yes Open
1190 54.308276283244666 -0.503734 -15.1619 2 13 7 0.88 1.00 - yes Open
1187 54.796057955280816 -0.525311 -16.6765 3 10 7 0.88 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.077kcal/mol
Ligand efficiency (LE) -0.4266kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.232
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 33HA

Physicochemical properties

Molecular weight 446.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.40
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 27.05kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 231.14kcal/mol
Minimised FF energy 204.10kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.