FAIRMol

OSA_Lib_234

Pose ID 48142 Compound 3334 Pose 1177

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.429 kcal/mol/HA) ✓ Good fit quality (FQ -4.30) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (30.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-14.599
kcal/mol
LE
-0.429
kcal/mol/HA
Fit Quality
-4.30
FQ (Leeson)
HAC
34
heavy atoms
MW
461
Da
LogP
1.79
cLogP
Strain ΔE
30.3 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 9 π–π 1 Clashes 4 Severe clashes 0
Final rank53.701255935605595Score-14.5991
Inter norm-0.455485Intra norm0.026099
Top1000noExcludedno
Contacts13H-bonds3
Artifact reasongeometry warning; 13 clashes; 4 protein contact clashes
ResiduesA:GLU466;A:GLU467;A:HIS461;A:LEU399;A:MET400;A:PHE396;A:PRO398;A:PRO462;A:SER394;A:SER395;A:SER464;A:SER470;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap6Native recall0.75
Jaccard0.40RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1184 3.6790895405749158 -0.404593 -13.2469 3 11 5 0.62 1.00 - no Open
1182 3.8450624526972663 -0.480145 -15.1588 3 11 5 0.62 1.00 - no Open
1181 3.934429235491084 -0.519206 -15.8686 3 12 6 0.75 1.00 - no Open
1176 4.074314858025007 -0.417412 -12.4101 2 8 5 0.62 1.00 - no Open
1172 4.555337198920386 -0.474056 -14.5695 3 13 8 1.00 1.00 - no Open
1170 5.062159442452728 -0.517066 -12.157 2 12 7 0.88 0.00 - no Open
1183 53.14433582047972 -0.423363 -13.1718 3 12 6 0.75 1.00 - no Open
1178 53.28995445794268 -0.457012 -13.6934 4 12 6 0.75 1.00 - no Open
1169 53.42773115001939 -0.434853 -11.1311 3 11 5 0.62 1.00 - no Open
1177 53.701255935605595 -0.455485 -14.5991 3 13 6 0.75 1.00 - no Current
1173 53.91230511494845 -0.440847 -11.975 4 10 4 0.50 1.00 - no Open
1171 54.41013456055068 -0.502946 -15.6489 2 12 7 0.88 1.00 - no Open
1175 54.80358110812957 -0.467986 -14.9226 2 12 7 0.88 1.00 - no Open
1174 55.08541691191576 -0.466314 -13.5165 2 11 7 0.88 0.00 - no Open
1180 55.402555293754595 -0.512896 -14.1834 2 11 7 0.88 0.00 - no Open
1179 55.17346273344424 -0.437713 -8.96343 4 11 4 0.50 1.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.599kcal/mol
Ligand efficiency (LE) -0.4294kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.296
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 34HA

Physicochemical properties

Molecular weight 460.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.79
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 30.29kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 231.31kcal/mol
Minimised FF energy 201.01kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.