FAIRMol

OSA_Lib_224

Pose ID 48112 Compound 3363 Pose 1147

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.451 kcal/mol/HA) ✓ Good fit quality (FQ -4.65) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (28.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-17.129
kcal/mol
LE
-0.451
kcal/mol/HA
Fit Quality
-4.65
FQ (Leeson)
HAC
38
heavy atoms
MW
518
Da
LogP
0.25
cLogP
Strain ΔE
28.5 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 23 π–π 2 Clashes 4 Severe clashes 0
Final rank54.78362369806652Score-17.1291
Inter norm-0.501957Intra norm0.0511902
Top1000noExcludedno
Contacts11H-bonds3
Artifact reasongeometry warning; 19 clashes; 4 protein contact clashes
ResiduesA:ASN402;A:GLU467;A:HIS461;A:LEU399;A:MET400;A:PHE396;A:PRO398;A:SER394;A:SER464;A:THR397;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap7Native recall0.88
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1149 4.380420581289307 -0.344785 -15.2196 4 12 6 0.75 1.00 - no Open
1148 4.628547783355802 -0.457194 -17.8303 2 12 6 0.75 1.00 - no Open
1151 4.963165621690814 -0.419739 -17.5342 2 10 7 0.88 0.00 - no Open
1141 5.3091933013882855 -0.367715 -13.2389 1 11 8 1.00 0.00 - no Open
1143 5.745868794151157 -0.34062 -11.9155 2 9 6 0.75 0.00 - no Open
1140 6.894579229847878 -0.576318 -13.427 2 14 8 1.00 0.00 - no Open
1145 54.44659666127433 -0.406132 -15.2873 2 11 7 0.88 0.00 - no Open
1139 54.76151659624603 -0.36092 -12.7766 1 11 7 0.88 0.00 - no Open
1147 54.78362369806652 -0.501957 -17.1291 3 11 7 0.88 0.00 - no Current
1144 55.351306427199106 -0.359925 -12.987 3 11 6 0.75 1.00 - no Open
1152 55.972734844709 -0.39102 -15.6819 3 13 8 1.00 0.00 - yes Open
1137 56.368601764642726 -0.349599 -13.3296 2 12 5 0.62 0.00 - yes Open
1138 56.53987961460191 -0.375221 -14.4577 2 13 7 0.88 0.00 - yes Open
1146 56.622673781036085 -0.453095 -15.7328 3 10 7 0.88 0.00 - yes Open
1150 57.389138968832604 -0.429198 -15.6252 3 13 8 1.00 0.00 - yes Open
1142 58.15632422365852 -0.429976 -14.7744 2 9 7 0.88 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -17.129kcal/mol
Ligand efficiency (LE) -0.4508kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.647
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 38HA

Physicochemical properties

Molecular weight 517.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.25
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 28.46kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 261.15kcal/mol
Minimised FF energy 232.69kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.