FAIRMol

OSA_Lib_185

Pose ID 48049 Compound 639 Pose 1084

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.383 kcal/mol/HA) ✓ Good fit quality (FQ -3.95) ✗ Very high strain energy (29.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-14.563
kcal/mol
LE
-0.383
kcal/mol/HA
Fit Quality
-3.95
FQ (Leeson)
HAC
38
heavy atoms
MW
517
Da
LogP
1.88
cLogP
Strain ΔE
29.8 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 10 π–π 0 Clashes 4 Severe clashes 0 ⚠ Hydrophobic exposure 48%
⚠️Partial hydrophobic solvent exposure
48% of hydrophobic surface appears solvent-exposed (16/33 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 33 Buried (contacted) 17 Exposed 16 LogP 1.88 H-bonds 2
Exposed fragments: phenyl (4/6 atoms exposed)phenyl (5/6 atoms exposed)phenyl (6/6 atoms exposed)aliphatic chain/group (1 atom exposed)
Final rank55.00743541524278Score-14.5629
Inter norm-0.432147Intra norm0.0489117
Top1000noExcludedno
Contacts12H-bonds2
Artifact reasongeometry warning; 20 clashes; 4 protein contact clashes
ResiduesA:GLU466;A:GLU467;A:HIS461;A:LEU399;A:MET393;A:MET400;A:PHE396;A:PRO398;A:SER394;A:SER395;A:SER470;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap6Native recall0.75
Jaccard0.43RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1087 4.3225639031029095 -0.469067 -15.5351 2 12 6 0.75 1.00 - no Open
1682 4.822428782793232 -0.574973 -20.0078 0 18 0 0.00 0.00 - no Open
1086 5.101010899152662 -0.371815 -12.4097 1 13 7 0.88 0.00 - no Open
1295 5.39625897207715 -0.573677 -19.4394 1 19 0 0.00 0.00 - no Open
1081 5.58153289922701 -0.390228 -16.9009 2 14 6 0.75 1.00 - no Open
1683 6.25042891583922 -0.632302 -24.5332 1 15 0 0.00 0.00 - no Open
1681 6.668996345435847 -0.58732 -20.2461 1 16 0 0.00 0.00 - no Open
1293 7.0457761337255125 -0.617927 -20.7888 0 22 0 0.00 0.00 - no Open
1290 8.325171038175231 -0.602483 -21.9589 1 19 0 0.00 0.00 - no Open
1088 54.635239060174506 -0.327996 -12.1045 3 14 6 0.75 1.00 - no Open
1083 54.65827673669226 -0.398049 -12.2755 3 13 8 1.00 0.00 - no Open
1084 55.00743541524278 -0.432147 -14.5629 2 12 6 0.75 1.00 - no Current
1082 55.03045979470512 -0.479943 -17.464 2 12 7 0.88 0.00 - no Open
1679 55.231811450195046 -0.491455 -18.9609 1 16 0 0.00 0.00 - no Open
1680 55.946621095636715 -0.494738 -15.8783 1 17 0 0.00 0.00 - no Open
1677 56.948725080742264 -0.609203 -20.8517 3 16 0 0.00 0.00 - no Open
1292 55.72704045128034 -0.582274 -22.0607 0 14 0 0.00 0.00 - yes Open
1085 55.89650249869848 -0.36287 -11.9186 3 16 8 1.00 0.00 - yes Open
1678 56.04238587597847 -0.732998 -25.1507 4 17 0 0.00 0.00 - yes Open
1289 57.50156813780052 -0.664958 -26.7266 1 17 0 0.00 0.00 - yes Open
1676 57.83556884909578 -0.588264 -25.1347 2 17 0 0.00 0.00 - yes Open
1296 57.85165481072552 -0.569824 -17.2283 1 19 0 0.00 0.00 - yes Open
1291 58.29120286658544 -0.589616 -19.5994 1 14 0 0.00 0.00 - yes Open
1294 60.273316324365645 -0.58113 -21.5496 1 12 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.563kcal/mol
Ligand efficiency (LE) -0.3832kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.951
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 38HA

Physicochemical properties

Molecular weight 516.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.88
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.81kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 157.45kcal/mol
Minimised FF energy 127.64kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.