FAIRMol

OSA_Lib_183

Pose ID 48024 Compound 677 Pose 1059

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good LE (-0.386 kcal/mol/HA) ✓ Good fit quality (FQ -3.95) ✓ Good H-bonds (3 bonds) ✗ Very high strain energy (37.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-14.278
kcal/mol
LE
-0.386
kcal/mol/HA
Fit Quality
-3.95
FQ (Leeson)
HAC
37
heavy atoms
MW
503
Da
LogP
1.88
cLogP
Strain ΔE
37.3 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 12 π–π 1 Clashes 4 Severe clashes 0
Final rank6.801132598817804Score-14.278
Inter norm-0.42519Intra norm0.0392969
Top1000noExcludedno
Contacts14H-bonds3
Artifact reasongeometry warning; 20 clashes; 4 protein contact clashes; high strain Δ 41.9
ResiduesA:GLU466;A:GLU467;A:HIS461;A:LEU399;A:MET393;A:MET400;A:PHE396;A:PRO398;A:PRO462;A:SER394;A:SER395;A:SER464;A:SER470;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap6Native recall0.75
Jaccard0.38RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1072 5.959432675645626 -0.340547 -13.2017 3 7 5 0.62 0.00 - no Open
1256 5.964710959533734 -0.632258 -18.974 0 22 0 0.00 0.00 - no Open
1064 6.001771173684105 -0.412686 -8.99484 2 10 6 0.75 0.00 - no Open
1255 6.1959168401841325 -0.659472 -21.2447 2 18 0 0.00 0.00 - no Open
1057 6.346866392093182 -0.41867 -12.1947 4 14 6 0.75 1.00 - no Open
1263 6.60231951508549 -0.683509 -25.6179 1 21 0 0.00 0.00 - no Open
1059 6.801132598817804 -0.42519 -14.278 3 14 6 0.75 1.00 - no Current
1254 6.867978178876968 -0.604759 -20.4945 2 16 0 0.00 0.00 - no Open
1260 7.197183510839782 -0.683727 -23.4348 1 14 0 0.00 0.00 - no Open
1253 54.41658892825658 -0.644899 -19.8124 0 20 0 0.00 0.00 - no Open
1060 55.306999765854236 -0.40253 -12.7252 3 12 7 0.88 0.00 - no Open
1250 55.6580625884546 -0.708155 -20.1601 1 21 0 0.00 0.00 - no Open
1259 7.038530585043578 -0.638988 -20.4351 1 17 0 0.00 0.00 - yes Open
1066 7.327863811853032 -0.56779 -20.2954 4 11 7 0.88 0.00 - yes Open
1069 7.340473730425458 -0.444895 -16.0066 4 11 6 0.75 0.00 - yes Open
1062 55.734685661358725 -0.381212 -15.1797 3 10 4 0.50 1.00 - yes Open
1252 55.974526153907696 -0.608194 -20.807 0 18 0 0.00 0.00 - yes Open
1251 56.7005535894911 -0.609644 -24.1202 0 12 0 0.00 0.00 - yes Open
1071 56.852117895408774 -0.5053 -14.5879 3 10 7 0.88 0.00 - yes Open
1070 56.902392631427915 -0.427454 -12.5198 3 9 6 0.75 0.00 - yes Open
1058 57.053999238947455 -0.531407 -16.739 3 10 7 0.88 0.00 - yes Open
1063 57.27490441539605 -0.52151 -16.4534 2 11 7 0.88 0.00 - yes Open
1065 57.402135370428766 -0.395583 -16.195 3 12 6 0.75 0.00 - yes Open
1262 57.40752138557653 -0.566931 -14.0268 1 20 0 0.00 0.00 - yes Open
1068 57.47314862622848 -0.582036 -20.6788 3 10 7 0.88 0.00 - yes Open
1067 57.54216830387588 -0.498979 -16.8833 4 9 5 0.62 0.00 - yes Open
1249 57.60690076970691 -0.621821 -21.5933 1 17 0 0.00 0.00 - yes Open
1258 57.7510495364424 -0.763052 -26.8159 1 20 0 0.00 0.00 - yes Open
1261 58.140804665646584 -0.620636 -19.3397 2 17 0 0.00 0.00 - yes Open
1061 58.444331624613994 -0.374921 -12.67 3 11 7 0.88 0.00 - yes Open
1257 58.58113556517499 -0.59477 -21.6424 1 17 0 0.00 0.00 - yes Open
1264 58.7524435649665 -0.781797 -26.637 2 19 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.278kcal/mol
Ligand efficiency (LE) -0.3859kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.951
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 502.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.88
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 37.25kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 149.06kcal/mol
Minimised FF energy 111.81kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.