FAIRMol

OSA_Lib_21

Pose ID 47783 Compound 3360 Pose 818

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.427 kcal/mol/HA) ✓ Good fit quality (FQ -4.37) ✗ Very high strain energy (25.7 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-15.784
kcal/mol
LE
-0.427
kcal/mol/HA
Fit Quality
-4.37
FQ (Leeson)
HAC
37
heavy atoms
MW
502
Da
LogP
2.91
cLogP
Strain ΔE
25.7 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 9 π–π 0 Clashes 2 Severe clashes 0 ⚠ Hydrophobic exposure 46%
⚠️Partial hydrophobic solvent exposure
47% of hydrophobic surface appears solvent-exposed (15/32 atoms). Partial exposure is common but may limit selectivity and membrane permeability.
Non-polar atoms 32 Buried (contacted) 17 Exposed 15 LogP 2.91 H-bonds 2
Exposed fragments: phenyl (6/6 atoms exposed)phenyl (6/6 atoms exposed)aliphatic chain/group (3 atoms exposed)
Final rank4.334055767654448Score-15.7838
Inter norm-0.400838Intra norm-0.0257524
Top1000noExcludedno
Contacts13H-bonds2
Artifact reasongeometry warning; 14 clashes; 2 protein contact clashes; high strain Δ 33.0
ResiduesA:GLU466;A:GLU467;A:HIS461;A:LEU399;A:MET400;A:PHE396;A:PRO398;A:PRO462;A:SER394;A:SER395;A:SER464;A:SER470;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap6Native recall0.75
Jaccard0.40RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
818 4.334055767654448 -0.400838 -15.7838 2 13 6 0.75 1.00 - no Current
819 4.458765365284852 -0.361306 -13.4756 2 14 8 1.00 1.00 - no Open
817 4.697065193936815 -0.386897 -14.2773 2 10 5 0.62 1.00 - no Open
806 4.895129712041564 -0.45368 -17.1294 2 13 7 0.88 1.00 - no Open
809 5.325353534483452 -0.469172 -18.392 3 12 7 0.88 0.00 - no Open
805 5.4775496321168635 -0.430721 -17.4508 3 13 7 0.88 1.00 - no Open
804 53.67538422447687 -0.49964 -15.5715 2 12 7 0.88 1.00 - no Open
810 53.700580361685034 -0.469246 -16.4261 2 12 6 0.75 1.00 - no Open
815 53.89692428958918 -0.383642 -13.7993 2 12 7 0.88 0.00 - no Open
814 54.03799527984407 -0.506004 -15.3056 3 11 7 0.88 0.00 - no Open
812 54.176280369546426 -0.449082 -16.9722 4 10 5 0.62 0.00 - no Open
813 54.653517013824256 -0.404507 -15.6536 3 8 5 0.62 0.00 - no Open
811 55.06101472748635 -0.46506 -14.4093 3 13 6 0.75 1.00 - no Open
808 55.35957025009879 -0.374323 -13.5829 3 11 5 0.62 0.00 - no Open
807 55.32786280317548 -0.579961 -16.4144 3 13 8 1.00 0.00 - yes Open
816 58.435001912920086 -0.420743 -12.1343 2 15 8 1.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -15.784kcal/mol
Ligand efficiency (LE) -0.4266kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.367
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 501.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.91
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 25.72kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 134.61kcal/mol
Minimised FF energy 108.89kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.