FAIRMol

KB_Leish_1

Pose ID 47555 Compound 2936 Pose 590

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.403 kcal/mol/HA) ✓ Good fit quality (FQ -3.92) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (29.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-12.485
kcal/mol
LE
-0.403
kcal/mol/HA
Fit Quality
-3.92
FQ (Leeson)
HAC
31
heavy atoms
MW
463
Da
LogP
5.31
cLogP
Strain ΔE
29.3 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 13 π–π 1 Clashes 4 Severe clashes 0
Final rank5.058545229338493Score-12.4848
Inter norm-0.495512Intra norm0.0927763
Top1000noExcludedno
Contacts10H-bonds4
Artifact reasongeometry warning; 12 clashes; 4 protein contact clashes; high strain Δ 39.5
ResiduesA:ASN402;A:GLU466;A:GLU467;A:HIS461;A:LEU399;A:PHE396;A:PRO398;A:SER464;A:THR397;A:THR463

Protein summary

492 residues
Protein targetT20Atoms7539
Residues492Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name9IFHContacts8
PoseOpen native poseH-bonds2
IFP residuesA:ASN402; A:GLU467; A:LEU399; A:PHE396; A:PRO398; A:SER394; A:SER470; A:THR397
Current overlap6Native recall0.75
Jaccard0.50RMSD-
H-bond strict1Strict recall0.50
H-bond same residue+role1Role recall1.00
H-bond same residue1Residue recall1.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
603 3.8044852916316727 -0.64201 -20.5404 5 16 7 0.88 1.00 - no Open
586 4.133639480999813 -0.459657 -14.3137 2 13 7 0.88 1.00 - no Open
606 4.35679852248012 -0.482688 -12.5267 3 10 6 0.75 1.00 - no Open
588 4.768513570953907 -0.486377 -11.4717 2 14 7 0.88 0.00 - no Open
604 4.897872850082145 -0.647312 -17.7174 3 13 5 0.62 1.00 - no Open
386 5.04889500330964 -0.582249 -15.3502 3 13 0 0.00 0.00 - no Open
590 5.058545229338493 -0.495512 -12.4848 4 10 6 0.75 1.00 - no Current
388 6.699680434476487 -0.876173 -23.3192 5 14 0 0.00 0.00 - no Open
392 7.357133203943192 -0.60999 -13.2463 4 12 0 0.00 0.00 - no Open
595 53.63205230972664 -0.576969 -14.0648 4 11 8 1.00 1.00 - no Open
598 53.823562632082904 -0.489728 -15.4323 2 11 5 0.62 1.00 - no Open
593 53.951856578686 -0.514805 -12.1895 2 13 7 0.88 0.00 - no Open
592 54.34499684632277 -0.508151 -16.6176 2 13 7 0.88 1.00 - no Open
608 54.48600947378974 -0.486729 -12.6698 2 12 6 0.75 1.00 - no Open
591 54.6487906993372 -0.458473 -13.1069 4 9 5 0.62 0.00 - no Open
380 6.995481301245248 -0.553748 -11.4268 2 17 0 0.00 0.00 - yes Open
383 7.493309597392498 -0.60514 -14.0984 3 13 0 0.00 0.00 - yes Open
378 7.5527008820243635 -0.642283 -15.0328 5 15 0 0.00 0.00 - yes Open
594 54.636622114209594 -0.539596 -17.8162 4 11 5 0.62 1.00 - yes Open
597 54.994155520595946 -0.541822 -15.8613 2 10 6 0.75 0.00 - yes Open
605 55.00188070827766 -0.533242 -15.8009 3 12 7 0.88 1.00 - yes Open
607 55.18067594788496 -0.538428 -16.8563 2 14 7 0.88 1.00 - yes Open
587 55.373123738271175 -0.51175 -14.9857 4 9 7 0.88 1.00 - yes Open
395 55.53515338651712 -0.606552 -15.425 1 14 0 0.00 0.00 - yes Open
585 55.59791610234486 -0.54959 -14.884 3 10 8 1.00 1.00 - yes Open
596 55.86089068647122 -0.538897 -15.7883 2 12 8 1.00 0.00 - yes Open
601 56.07350512110974 -0.564946 -13.7397 2 12 8 1.00 1.00 - yes Open
589 56.121280930227165 -0.56093 -12.5425 2 12 7 0.88 0.00 - yes Open
600 56.23209528423411 -0.541966 -18.3447 3 10 7 0.88 0.00 - yes Open
393 56.23572476535945 -0.683482 -17.0219 3 15 0 0.00 0.00 - yes Open
602 56.32772230499301 -0.49774 -16.9141 5 9 4 0.50 1.00 - yes Open
379 56.6266773907136 -0.547826 -9.18538 2 15 0 0.00 0.00 - yes Open
385 56.70770719150399 -0.731306 -23.6734 3 13 0 0.00 0.00 - yes Open
381 56.88766429102111 -0.810642 -23.3319 3 15 0 0.00 0.00 - yes Open
387 56.91839106122524 -0.714746 -20.9139 2 16 0 0.00 0.00 - yes Open
391 57.01029957077979 -0.717756 -20.4792 6 10 0 0.00 0.00 - yes Open
389 57.14245644007512 -0.769954 -19.345 5 15 0 0.00 0.00 - yes Open
384 57.419456380965755 -0.588605 -14.6981 2 16 0 0.00 0.00 - yes Open
376 57.764354561242754 -0.543591 -15.164 2 10 0 0.00 0.00 - yes Open
382 57.79014964446977 -0.736543 -22.5192 3 15 0 0.00 0.00 - yes Open
390 57.809059650181844 -0.771028 -23.1672 5 14 0 0.00 0.00 - yes Open
397 57.90883832160699 -0.617507 -18.4212 2 14 0 0.00 0.00 - yes Open
398 57.984342221875046 -0.83277 -24.6131 3 15 0 0.00 0.00 - yes Open
377 58.19397974886769 -0.658949 -17.5313 2 14 0 0.00 0.00 - yes Open
394 58.19821300993624 -0.766089 -23.6755 3 14 0 0.00 0.00 - yes Open
599 58.35248215172916 -0.515234 -15.3395 3 8 6 0.75 0.00 - yes Open
396 60.01756934145726 -0.677641 -19.8411 4 11 0 0.00 0.00 - yes Open
399 61.76318792298458 -0.634659 -17.3185 4 11 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -12.485kcal/mol
Ligand efficiency (LE) -0.4027kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -3.924
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 463.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.31
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.28kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 100.22kcal/mol
Minimised FF energy 70.94kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.