FAIRMol

Z49732247

Pose ID 46864 Compound 2028 Pose 2131

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.361 kcal/mol/HA) ✓ Good fit quality (FQ -12.02) ✓ Strong H-bond network (11 bonds) ✗ High strain energy (12.5 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-31.314
kcal/mol
LE
-1.361
kcal/mol/HA
Fit Quality
-12.02
FQ (Leeson)
HAC
23
heavy atoms
MW
311
Da
LogP
1.70
cLogP
Strain ΔE
12.5 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 11 Hydrophobic 14 π–π 0 Clashes 5 Severe clashes 0
Final rank3.3500909879271155Score-31.3137
Inter norm-1.26361Intra norm-0.120386
Top1000noExcludedno
Contacts15H-bonds11
Artifact reasongeometry warning; 14 clashes; 5 protein contact clashes; moderate strain Δ 13.3
ResiduesC:ARG287;C:ASP327;C:CYS52;C:CYS57;C:GLY56;C:ILE199;C:LEU334;C:LYS60;C:MET333;C:NDP800;C:PHE367;C:SER14;C:SER162;C:THR335;C:THR51

Protein summary

493 residues
Protein targetT19Atoms7541
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:330; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name2WOVContacts27
PoseOpen native poseH-bonds16
IFP residuesC:ALA284; C:ALA365; C:ARG222; C:ARG228; C:ARG287; C:ASN223; C:ASN254; C:GLN165; C:GLU202; C:GLY195; C:GLY196; C:GLY197; C:GLY286; C:ILE199; C:ILE285; C:LEU227; C:LEU334; C:LYS60; C:MET333; C:NDP800; C:PHE198; C:PHE367; C:PRO167; C:SER200; C:TYR221; C:VAL194; C:VAL366
Current overlap7Native recall0.26
Jaccard0.20RMSD-
H-bond strict1Strict recall0.08
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.25

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
2494 2.5582396215047405 -0.931924 -19.4442 7 14 0 0.00 0.00 - no Open
2131 3.3500909879271155 -1.26361 -31.3137 11 15 7 0.26 0.20 - no Current
2127 3.450789308807371 -1.37194 -33.0595 10 16 7 0.26 0.20 - no Open
2129 3.79862132008788 -1.10687 -27.4074 10 15 7 0.26 0.20 - no Open
2133 4.263918140872896 -1.30626 -29.8803 10 16 7 0.26 0.20 - no Open
2489 4.317854091732456 -1.22574 -25.6178 6 18 0 0.00 0.00 - no Open
2622 4.801894368066783 -0.755595 -18.745 10 6 0 0.00 0.00 - no Open
2490 7.000237443658768 -1.00542 -25.4149 8 13 0 0.00 0.00 - yes Open
2627 7.228723845451232 -1.06665 -24.7818 13 14 0 0.00 0.00 - yes Open
2128 7.677396800391303 -1.44534 -28.4543 7 18 8 0.30 0.20 - yes Open
2628 7.749323051501671 -0.751957 -18.6197 9 5 0 0.00 0.00 - yes Open
2492 7.760626518140129 -0.949545 -24.1796 8 12 0 0.00 0.00 - yes Open
2626 7.964704120100794 -0.696659 -13.9958 9 9 0 0.00 0.00 - yes Open
2623 8.219116212124502 -1.08553 -22.761 14 14 0 0.00 0.00 - yes Open
2126 8.737107733756439 -1.52382 -26.7145 10 17 7 0.26 0.20 - yes Open
2132 8.741610438820343 -1.46076 -26.721 9 18 8 0.30 0.20 - yes Open
2493 9.153896896196803 -1.02599 -21.8038 12 16 0 0.00 0.00 - yes Open
2625 9.272227844688931 -1.11233 -23.8024 12 14 0 0.00 0.00 - yes Open
2130 9.768135939683326 -1.40066 -25.1442 8 16 7 0.26 0.20 - yes Open
2624 9.79400155185025 -0.678171 -17.2739 9 8 0 0.00 0.00 - yes Open
2621 10.130550327031907 -1.14839 -23.4369 14 15 0 0.00 0.00 - yes Open
2491 10.18841919495861 -1.16694 -23.0743 13 15 0 0.00 0.00 - yes Open
2487 10.558774742673078 -1.2773 -27.7269 12 17 0 0.00 0.00 - yes Open
2488 11.656258305698623 -1.09487 -25.8121 7 16 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -31.314kcal/mol
Ligand efficiency (LE) -1.3615kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -12.016
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 23HA

Physicochemical properties

Molecular weight 311.3Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.70
Lipinski: ≤ 5
Rotatable bonds 2

Conformational strain (MMFF94s)

Strain energy (ΔE) 12.49kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 89.72kcal/mol
Minimised FF energy 77.23kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.