FAIRMol

Z19696461

Pose ID 46628 Compound 987 Pose 1895

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-1.222 kcal/mol/HA) ✓ Good fit quality (FQ -11.11) ✓ Good H-bonds (5 bonds) ✗ High strain energy (10.6 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-30.561
kcal/mol
LE
-1.222
kcal/mol/HA
Fit Quality
-11.11
FQ (Leeson)
HAC
25
heavy atoms
MW
352
Da
LogP
2.97
cLogP
Strain ΔE
10.6 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 15 π–π 1 Clashes 12 Severe clashes 0
Final rank5.046651469343701Score-30.5605
Inter norm-1.27119Intra norm0.0441311
Top1000noExcludedno
Contacts15H-bonds5
Artifact reasongeometry warning; 12 clashes; 12 protein contact clashes
ResiduesC:ALA365;C:CYS57;C:GLU436;C:GLY56;C:ILE438;C:LEU334;C:LYS60;C:MET333;C:NDP800;C:PHE367;C:PRO336;C:PRO435;C:SER364;C:THR335;C:THR51

Protein summary

493 residues
Protein targetT19Atoms7541
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:330; TYR:294; ASP:264; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name2WOVContacts27
PoseOpen native poseH-bonds16
IFP residuesC:ALA284; C:ALA365; C:ARG222; C:ARG228; C:ARG287; C:ASN223; C:ASN254; C:GLN165; C:GLU202; C:GLY195; C:GLY196; C:GLY197; C:GLY286; C:ILE199; C:ILE285; C:LEU227; C:LEU334; C:LYS60; C:MET333; C:NDP800; C:PHE198; C:PHE367; C:PRO167; C:SER200; C:TYR221; C:VAL194; C:VAL366
Current overlap6Native recall0.22
Jaccard0.17RMSD-
H-bond strict1Strict recall0.08
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.25

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1895 5.046651469343701 -1.27119 -30.5605 5 15 6 0.22 0.20 - no Current
1771 5.408155498072421 -0.851318 -18.8784 3 10 0 0.00 0.00 - no Open
1770 5.2377549899797815 -0.961165 -24.027 4 13 0 0.00 0.00 - yes Open
1896 9.605669122289578 -1.20937 -19.9274 10 17 8 0.30 0.40 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -30.561kcal/mol
Ligand efficiency (LE) -1.2224kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -11.113
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 25HA

Physicochemical properties

Molecular weight 352.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.97
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 10.55kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 10.28kcal/mol
Minimised FF energy -0.28kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.