FAIRMol

OSA_Lib_184

Pose ID 4584 Compound 611 Pose 1266

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.566 kcal/mol/HA) ✓ Good fit quality (FQ -5.76) ✗ Very high strain energy (31.2 kcal/mol) ✗ No H-bonds detected ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.386
kcal/mol
LE
-0.566
kcal/mol/HA
Fit Quality
-5.76
FQ (Leeson)
HAC
36
heavy atoms
MW
491
Da
LogP
1.74
cLogP
Strain ΔE
31.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 31.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 0 Hydrophobic 24 π–π 0 Clashes 3 Severe clashes 0
Final rank5.916219393702416Score-20.3863
Inter norm-0.505792Intra norm-0.0604948
Top1000noExcludedno
Contacts21H-bonds0
Artifact reasongeometry warning; 17 clashes; 3 protein contact clashes; high strain Δ 41.9
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR180;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.71RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

No hydrogen bonds detected for this pose.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1277 4.955390243682244 -0.633304 -23.2003 1 20 16 0.80 0.00 - no Open
1284 5.266590438213333 -0.589116 -20.5555 0 21 16 0.80 0.00 - no Open
1273 5.420218368573264 -0.69434 -23.3365 1 17 13 0.65 0.00 - no Open
1276 5.63123130661502 -0.577185 -19.3035 0 23 18 0.90 0.00 - no Open
1266 5.916219393702416 -0.505792 -20.3863 0 21 17 0.85 0.00 - no Current
1268 6.237408435825435 -0.504901 -16.749 0 20 16 0.80 0.00 - no Open
1271 6.677440558013149 -0.671078 -20.2642 0 21 17 0.85 0.00 - no Open
1282 7.103710860788376 -0.529393 -16.305 1 19 15 0.75 0.00 - no Open
1283 8.149754730529782 -0.703227 -24.5366 0 22 19 0.95 0.00 - no Open
1272 55.168442638495705 -0.597273 -19.3811 1 17 16 0.80 0.00 - no Open
1267 55.22585166049036 -0.722343 -24.5284 1 20 16 0.80 0.00 - no Open
1278 55.34802207569263 -0.59464 -20.3427 0 20 17 0.85 0.00 - no Open
1274 55.90467238694108 -0.577796 -19.3768 1 15 14 0.70 0.00 - no Open
1279 55.15930333170979 -0.54678 -18.2212 0 20 17 0.85 0.00 - yes Open
1269 55.430613126236565 -0.56603 -20.9268 0 20 17 0.85 0.00 - yes Open
1286 55.94254527420868 -0.723334 -26.5795 1 20 16 0.80 0.00 - yes Open
1275 56.10591493197533 -0.739461 -28.2783 1 21 17 0.85 0.00 - yes Open
1288 56.22278985082605 -0.484989 -14.9191 0 16 15 0.75 0.00 - yes Open
1281 56.69113764342162 -0.65413 -21.5281 2 17 16 0.80 0.20 - yes Open
1287 56.77900350542991 -0.639226 -21.8545 1 20 17 0.85 0.00 - yes Open
1285 57.09888257553469 -0.639662 -22.3896 1 18 15 0.75 0.00 - yes Open
1270 57.15492175021484 -0.704798 -28.3287 1 20 16 0.80 0.00 - yes Open
1265 57.22681303945254 -0.593801 -19.0446 2 16 15 0.75 0.20 - yes Open
1280 57.580035907571485 -0.481053 -17.2959 0 16 12 0.60 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.386kcal/mol
Ligand efficiency (LE) -0.5663kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.756
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 36HA

Physicochemical properties

Molecular weight 490.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.74
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 31.22kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 188.43kcal/mol
Minimised FF energy 157.21kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.