FAIRMol

Z57907181

Pose ID 43924 Compound 1661 Pose 1837

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.627 kcal/mol/HA) ✓ Good fit quality (FQ -6.32) ✓ Strong H-bond network (7 bonds) ✗ Very high strain energy (22.0 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.941
kcal/mol
LE
-0.627
kcal/mol/HA
Fit Quality
-6.32
FQ (Leeson)
HAC
35
heavy atoms
MW
472
Da
LogP
4.29
cLogP
Strain ΔE
22.0 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 7 Hydrophobic 24 π–π 3 Clashes 7 Severe clashes 0
Final rank4.916841023503335Score-21.9414
Inter norm-0.613323Intra norm-0.0135737
Top1000noExcludedno
Contacts12H-bonds7
Artifact reasongeometry warning; 13 clashes; 7 protein contact clashes; high strain Δ 23.1
ResiduesA:ASP116;A:GLU18;A:GLY112;A:ILE106;A:ILE339;A:LEU17;A:MET113;A:SER109;A:SER14;A:THR117;A:TRP21;A:TYR110

Protein summary

493 residues
Protein targetT18Atoms7550
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts13
PoseOpen native poseH-bonds0
IFP residuesA:ASP116; A:GLU18; A:GLY112; A:ILE106; A:LEU17; A:MET113; A:SER109; A:THR117; A:THR335; A:TRP21; A:TYR110; A:VAL53; A:VAL58
Current overlap10Native recall0.77
Jaccard0.67RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1299 4.67666138086561 -0.800498 -22.8564 4 13 0 0.00 - - no Open
1383 4.8634702985950184 -0.710536 -19.5805 7 19 0 0.00 - - no Open
1385 4.897123544374696 -0.711011 -19.3654 7 18 0 0.00 - - no Open
1837 4.916841023503335 -0.613323 -21.9414 7 12 10 0.77 - - no Current
1873 6.014167817838366 -0.437553 -13.5507 4 10 0 0.00 - - no Open
1836 6.45394666125905 -0.550271 -16.7366 4 11 6 0.46 - - yes Open
1835 6.787346339305998 -0.500954 -13.4974 4 8 8 0.62 - - yes Open
1872 7.142668701095011 -0.429101 -13.6955 5 11 0 0.00 - - yes Open
1833 7.1564826313641445 -0.521505 -14.4645 5 11 8 0.62 - - yes Open
1838 7.2365799038806955 -0.497374 -18.02 6 10 8 0.62 - - yes Open
1871 7.261612866237191 -0.437793 -10.8721 5 10 0 0.00 - - yes Open
1870 7.361473628938555 -0.570175 -19.8317 8 14 0 0.00 - - yes Open
1302 7.509224060007598 -0.955819 -24.3858 6 17 0 0.00 - - yes Open
1834 7.732410263948414 -0.471613 -14.2802 4 12 7 0.54 - - yes Open
1304 7.997267095980302 -0.883007 -24.3786 6 18 0 0.00 - - yes Open
1387 8.06576320543421 -0.61579 -18.9134 9 18 0 0.00 - - yes Open
1298 8.29306536925217 -0.864988 -20.0465 5 17 0 0.00 - - yes Open
1388 8.350302464770216 -0.680049 -24.7454 11 17 0 0.00 - - yes Open
1874 8.37315139556177 -0.478477 -15.0134 7 8 0 0.00 - - yes Open
1297 8.4343591372871 -0.746478 -22.8458 5 14 0 0.00 - - yes Open
1869 8.833036889510451 -0.531912 -15.9374 7 13 0 0.00 - - yes Open
1384 10.987916074415484 -0.719643 -25.915 9 17 0 0.00 - - yes Open
1386 11.344449559314778 -0.705221 -26.3153 9 16 0 0.00 - - yes Open
1300 13.222307394321126 -0.907521 -29.2878 8 17 0 0.00 - - yes Open
1303 13.33420476304861 -0.76258 -20.501 7 16 0 0.00 - - yes Open
1301 14.805388367185293 -0.802401 -20.3129 7 16 0 0.00 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.941kcal/mol
Ligand efficiency (LE) -0.6269kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.323
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 471.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.29
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 21.97kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 118.36kcal/mol
Minimised FF energy 96.39kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.