FAIRMol

OSA_Lib_84

Pose ID 4374 Compound 347 Pose 1056

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.410 kcal/mol/HA) ✓ Good fit quality (FQ -4.14) ✗ Very high strain energy (29.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-14.352
kcal/mol
LE
-0.410
kcal/mol/HA
Fit Quality
-4.14
FQ (Leeson)
HAC
35
heavy atoms
MW
479
Da
LogP
1.59
cLogP
Strain ΔE
29.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 29.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 2 Clashes 10 Severe clashes 0
Final rank55.90140041925345Score-14.352
Inter norm-0.617017Intra norm0.206959
Top1000noExcludedno
Contacts16H-bonds2
Artifact reasongeometry warning; 17 clashes; 10 protein contact clashes
ResiduesA:ARG48;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:THR83;A:TRP47;A:VAL156;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap13Native recall0.65
Jaccard0.57RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1055 5.313328596878003 -0.612484 -18.9103 0 18 15 0.75 0.00 - no Open
1111 5.988282725291934 -0.570811 -8.07888 2 18 0 0.00 0.00 - no Open
1108 6.092297833020478 -0.655499 -18.069 1 19 0 0.00 0.00 - no Open
482 6.323120530680791 -0.579549 -19.2462 8 17 0 0.00 0.00 - no Open
1066 6.50554339869121 -0.661308 -16.3273 3 19 18 0.90 0.60 - no Open
1065 6.568253867525926 -0.611064 -15.647 2 19 14 0.70 0.20 - no Open
1054 6.713041137958088 -0.554606 -17.7904 3 20 16 0.80 0.00 - no Open
1048 6.85325019789474 -0.581063 -21.0538 0 15 12 0.60 0.00 - no Open
1068 7.1399807136827 -0.689684 -19.87 4 18 16 0.80 0.40 - no Open
1114 7.602068458155432 -0.596839 -14.0415 4 19 0 0.00 0.00 - no Open
475 7.802690905935957 -0.863376 -26.0776 11 18 0 0.00 0.00 - no Open
1063 55.62898232574176 -0.665917 -17.2122 0 20 16 0.80 0.00 - no Open
1056 55.90140041925345 -0.617017 -14.352 2 16 13 0.65 0.20 - no Current
1110 56.51773991033714 -0.619035 -21.0296 3 21 0 0.00 0.00 - no Open
1109 56.57259995587179 -0.531233 -8.34814 1 17 0 0.00 0.00 - no Open
1051 56.641776096054365 -0.746961 -20.3703 0 22 18 0.90 0.00 - no Open
1104 56.759070891457476 -0.666067 -19.5598 2 17 0 0.00 0.00 - no Open
494 7.058518467030137 -0.730332 -23.7163 9 15 0 0.00 0.00 - yes Open
489 7.505909064837407 -0.846 -28.4809 9 17 0 0.00 0.00 - yes Open
491 7.627376238736397 -0.803525 -23.8294 9 15 0 0.00 0.00 - yes Open
477 8.816182954140789 -0.857347 -12.5541 8 18 0 0.00 0.00 - yes Open
1107 56.159883063747614 -0.589322 -12.9484 0 21 0 0.00 0.00 - yes Open
472 56.24142153355094 -0.791382 -22.8879 7 18 0 0.00 0.00 - yes Open
1067 56.425855623370396 -0.788506 -22.0939 1 21 18 0.90 0.00 - yes Open
1101 56.53961540616086 -0.593157 -20.3236 3 21 0 0.00 0.00 - yes Open
1052 56.54367311783271 -0.667232 -14.1979 1 17 12 0.60 0.20 - yes Open
479 56.582124053825474 -0.746436 -18.3532 8 17 0 0.00 0.00 - yes Open
1062 56.7457335393394 -0.598921 -21.0503 1 13 9 0.45 0.00 - yes Open
1105 56.80164721567153 -0.581867 -18.3978 4 20 0 0.00 0.00 - yes Open
1103 56.80535482516133 -0.587925 -10.9579 2 16 0 0.00 0.00 - yes Open
1113 56.84804431874544 -0.584243 -21.7354 4 17 0 0.00 0.00 - yes Open
478 56.87215583759871 -0.688083 -23.3657 9 16 0 0.00 0.00 - yes Open
1060 56.88122770236947 -0.684093 -21.6167 2 15 11 0.55 0.20 - yes Open
488 56.92737903641403 -0.826983 -26.0155 8 17 0 0.00 0.00 - yes Open
486 57.03505156484431 -0.615421 -20.8054 8 17 0 0.00 0.00 - yes Open
1047 57.075008099644876 -0.629676 -17.8448 2 17 14 0.70 0.00 - yes Open
1046 57.253066991192924 -0.584392 -17.926 1 19 15 0.75 0.00 - yes Open
1112 57.28994090004693 -0.547133 -18.9455 5 19 0 0.00 0.00 - yes Open
476 57.30781031362373 -0.861047 -22.4843 8 17 0 0.00 0.00 - yes Open
1057 57.42933461016668 -0.547606 -15.8139 2 16 11 0.55 0.20 - yes Open
1064 57.56952935530013 -0.676322 -19.8317 1 18 16 0.80 0.20 - yes Open
1106 57.57225940358665 -0.610146 -17.3823 2 16 0 0.00 0.00 - yes Open
1102 57.72100554110568 -0.648471 -19.9743 1 19 0 0.00 0.00 - yes Open
1115 57.84458738283716 -0.697945 -18.3648 2 19 0 0.00 0.00 - yes Open
484 58.12728328618293 -0.579573 -17.9339 7 13 0 0.00 0.00 - yes Open
1059 58.14142217846666 -0.698779 -20.3778 2 21 18 0.90 0.00 - yes Open
1050 58.23071824909503 -0.723755 -21.8716 1 15 12 0.60 0.00 - yes Open
480 58.23380991509278 -0.578297 -16.1747 6 16 0 0.00 0.00 - yes Open
1045 58.360638563081004 -0.755706 -20.2963 5 18 16 0.80 0.40 - yes Open
1049 58.3822084194494 -0.594774 -22.2501 2 11 9 0.45 0.00 - yes Open
1061 58.68049224120255 -0.610465 -20.2738 2 17 13 0.65 0.20 - yes Open
1116 58.76421747856189 -0.583896 -15.9692 4 18 0 0.00 0.00 - yes Open
487 58.95863723810485 -0.504495 -10.2032 6 15 0 0.00 0.00 - yes Open
492 58.974693798442935 -0.774617 -22.1204 8 17 0 0.00 0.00 - yes Open
1058 59.12153058551491 -0.618346 -13.9963 3 16 13 0.65 0.20 - yes Open
483 59.12197035768773 -0.559579 -17.5314 4 14 0 0.00 0.00 - yes Open
473 59.172575797327 -0.781301 -24.6413 10 19 0 0.00 0.00 - yes Open
485 59.19387800585095 -0.592835 -17.5626 5 13 0 0.00 0.00 - yes Open
495 59.26072218810411 -0.747936 -9.85485 8 16 0 0.00 0.00 - yes Open
474 59.49695670503676 -0.779613 -23.305 8 19 0 0.00 0.00 - yes Open
490 59.68628364171217 -0.752681 -18.5042 8 15 0 0.00 0.00 - yes Open
493 60.34995577033395 -0.820578 -27.52 9 16 0 0.00 0.00 - yes Open
481 60.36685694644978 -0.601056 -19.1838 6 14 0 0.00 0.00 - yes Open
1053 64.16778935268795 -0.634539 -19.648 1 18 15 0.75 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.352kcal/mol
Ligand efficiency (LE) -0.4101kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.136
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 35HA

Physicochemical properties

Molecular weight 478.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.59
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 29.07kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 80.58kcal/mol
Minimised FF energy 51.51kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.