FAIRMol

NMT-TY0616

Pose ID 43515 Compound 170 Pose 1428

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.534 kcal/mol/HA) ✓ Good fit quality (FQ -5.04) ✓ Good H-bonds (5 bonds) ✗ Very high strain energy (44.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-14.947
kcal/mol
LE
-0.534
kcal/mol/HA
Fit Quality
-5.04
FQ (Leeson)
HAC
28
heavy atoms
MW
424
Da
LogP
2.15
cLogP
Strain ΔE
44.9 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 2 Clashes 3 Severe clashes 0
Final rank3.9298186005779687Score-14.9466
Inter norm-0.605853Intra norm0.0720444
Top1000noExcludedno
Contacts13H-bonds5
Artifact reasongeometry warning; 8 clashes; 3 protein contact clashes; high strain Δ 40.5
ResiduesA:CYS52;A:GLU18;A:GLY13;A:ILE339;A:LEU17;A:MET113;A:SER109;A:SER14;A:THR335;A:TRP21;A:TYR110;A:VAL53;A:VAL58

Protein summary

493 residues
Protein targetT18Atoms7550
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts13
PoseOpen native poseH-bonds0
IFP residuesA:ASP116; A:GLU18; A:GLY112; A:ILE106; A:LEU17; A:MET113; A:SER109; A:THR117; A:THR335; A:TRP21; A:TYR110; A:VAL53; A:VAL58
Current overlap9Native recall0.69
Jaccard0.53RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
684 2.998114427523072 -0.914312 -27.7045 0 14 0 0.00 - - no Open
683 3.423239363374118 -0.875663 -24.9781 2 14 0 0.00 - - no Open
1428 3.9298186005779687 -0.605853 -14.9466 5 13 9 0.69 - - no Current
1426 4.399758051131676 -0.71286 -18.2694 5 14 10 0.77 - - no Open
2143 4.422122670354982 -0.930092 -24.8423 3 19 0 0.00 - - no Open
1101 4.667749878403291 -0.757253 -20.6541 4 18 0 0.00 - - no Open
873 4.99792091193104 -0.804988 -21.6072 3 20 0 0.00 - - no Open
2876 5.155972220850824 -0.702132 -19.841 7 15 0 0.00 - - no Open
870 5.524561054711304 -0.782276 -19.8489 3 19 0 0.00 - - no Open
869 6.723600251274246 -0.830931 -22.6515 3 18 0 0.00 - - no Open
872 7.305716645891471 -0.837824 -22.3125 5 20 0 0.00 - - no Open
2875 4.806340784632896 -0.853624 -23.9239 4 16 0 0.00 - - yes Open
2144 6.839755713793148 -0.883202 -23.6779 3 18 0 0.00 - - yes Open
1102 6.922431059103933 -0.813433 -22.2882 11 14 0 0.00 - - yes Open
1098 7.199951055038816 -0.854857 -22.3935 9 15 0 0.00 - - yes Open
1099 7.644389496276355 -0.821841 -24.4138 6 12 0 0.00 - - yes Open
1429 7.695611950082826 -0.8002 -21.9823 8 14 9 0.69 - - yes Open
1100 7.749640710391436 -0.842191 -17.8741 3 19 0 0.00 - - yes Open
871 7.815700220262551 -0.786889 -13.9217 4 19 0 0.00 - - yes Open
868 8.1520816586295 -0.790344 -24.4174 5 19 0 0.00 - - yes Open
1427 8.345073488173243 -0.625804 -20.6871 5 13 7 0.54 - - yes Open
1103 9.503399408675296 -0.846508 -23.4398 1 17 0 0.00 - - yes Open
874 15.203640504046483 -0.795666 -22.1396 2 20 0 0.00 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -14.947kcal/mol
Ligand efficiency (LE) -0.5338kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.039
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 28HA

Physicochemical properties

Molecular weight 423.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.15
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 44.93kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 14.57kcal/mol
Minimised FF energy -30.36kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.