FAIRMol

OSA_Lib_81

Pose ID 4340 Compound 709 Pose 1022

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.691 kcal/mol/HA) ✓ Good fit quality (FQ -7.12) ✗ Very high strain energy (24.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-26.262
kcal/mol
LE
-0.691
kcal/mol/HA
Fit Quality
-7.12
FQ (Leeson)
HAC
38
heavy atoms
MW
518
Da
LogP
3.93
cLogP
Strain ΔE
24.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: mixed
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 24.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 7 Severe clashes 1
Final rank7.299943420607154Score-26.2625
Inter norm-0.653108Intra norm-0.03801
Top1000noExcludedyes
Contacts13H-bonds1
Artifact reasonexcluded; geometry warning; 17 clashes; 1 protein clash; high strain Δ 23.2
ResiduesA:ARG97;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:SER44;A:SER86;A:THR54

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap10Native recall0.50
Jaccard0.43RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1027 6.822704372144355 -0.624761 -17.7279 1 17 12 0.60 0.20 - no Open
1010 6.951751574540021 -0.646538 -25.7143 6 17 16 0.80 0.80 - no Open
1026 7.094287334300263 -0.639275 -23.7617 1 21 17 0.85 0.00 - no Open
1007 8.05176775701517 -0.647097 -23.4754 2 21 17 0.85 0.20 - no Open
1015 8.398258772771907 -0.521279 -14.9385 1 18 14 0.70 0.00 - no Open
1005 57.657619813151406 -0.630418 -20.2269 2 16 11 0.55 0.00 - no Open
1022 7.299943420607154 -0.653108 -26.2625 1 13 10 0.50 0.00 - yes Current
1009 55.805742056293134 -0.630072 -16.803 1 21 18 0.90 0.00 - yes Open
1014 56.2875781932553 -0.651308 -23.8815 1 14 11 0.55 0.00 - yes Open
1013 56.78374927155866 -0.598157 -16.2061 2 18 17 0.85 0.40 - yes Open
1028 56.90150959242682 -0.684463 -22.8726 1 22 17 0.85 0.00 - yes Open
1019 57.02520469114295 -0.686472 -24.0861 1 21 16 0.80 0.20 - yes Open
1012 57.15269072922803 -0.621102 -23.7081 2 16 14 0.70 0.00 - yes Open
1011 57.30563772090751 -0.605626 -21.6388 1 19 15 0.75 0.00 - yes Open
1025 57.758925345189866 -0.670238 -17.3409 4 18 16 0.80 0.20 - yes Open
1023 57.868460667105666 -0.651571 -23.6812 1 19 14 0.70 0.20 - yes Open
1020 58.34787606194498 -0.612191 -20.4774 0 22 16 0.80 0.00 - yes Open
1017 58.86457689985148 -0.614434 -20.1777 0 20 16 0.80 0.00 - yes Open
1008 59.888711794691346 -0.728931 -26.4351 4 20 17 0.85 0.40 - yes Open
1006 60.00789818717066 -0.629589 -22.342 1 14 12 0.60 0.00 - yes Open
1021 60.196004145692974 -0.63783 -27.1067 1 15 11 0.55 0.00 - yes Open
1016 61.003200045112486 -0.670707 -22.0919 0 15 13 0.65 0.00 - yes Open
1024 61.47334636016435 -0.774733 -28.3258 3 19 16 0.80 0.60 - yes Open
1018 63.28505917139624 -0.653678 -19.3117 1 20 16 0.80 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.262kcal/mol
Ligand efficiency (LE) -0.6911kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.125
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 38HA

Physicochemical properties

Molecular weight 517.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.93
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 24.53kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 57.45kcal/mol
Minimised FF energy 32.92kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.