FAIRMol

TC493

Pose ID 43324 Compound 3085 Pose 1237

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.659 kcal/mol/HA) ✓ Good fit quality (FQ -6.48) ✓ Good H-bonds (3 bonds) ✗ High strain energy (19.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.100
kcal/mol
LE
-0.659
kcal/mol/HA
Fit Quality
-6.48
FQ (Leeson)
HAC
32
heavy atoms
MW
443
Da
LogP
3.31
cLogP
Strain ΔE
19.9 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 3 Hydrophobic 24 π–π 0 Clashes 4 Severe clashes 0
Final rank3.4923915045259353Score-21.0999
Inter norm-0.659455Intra norm8.37005e-05
Top1000noExcludedno
Contacts13H-bonds3
Artifact reasongeometry warning; 12 clashes; 4 protein contact clashes; moderate strain Δ 18.4
ResiduesA:ASP116;A:GLU18;A:GLY13;A:GLY49;A:ILE339;A:LEU17;A:MET113;A:SER109;A:SER14;A:THR335;A:TRP21;A:TYR110;A:VAL53

Protein summary

493 residues
Protein targetT18Atoms7550
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts13
PoseOpen native poseH-bonds0
IFP residuesA:ASP116; A:GLU18; A:GLY112; A:ILE106; A:LEU17; A:MET113; A:SER109; A:THR117; A:THR335; A:TRP21; A:TYR110; A:VAL53; A:VAL58
Current overlap9Native recall0.69
Jaccard0.53RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1237 3.4923915045259353 -0.659455 -21.0999 3 13 9 0.69 - - no Current
1236 5.593806858404492 -0.671888 -24.5081 3 14 9 0.69 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.100kcal/mol
Ligand efficiency (LE) -0.6594kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.484
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 442.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.31
Lipinski: ≤ 5
Rotatable bonds 2

Conformational strain (MMFF94s)

Strain energy (ΔE) 19.95kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 124.14kcal/mol
Minimised FF energy 104.19kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.