FAIRMol

OSA_Lib_78

Pose ID 4309 Compound 631 Pose 991

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.581 kcal/mol/HA) ✓ Good fit quality (FQ -5.95) ✗ Very high strain energy (33.7 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-21.510
kcal/mol
LE
-0.581
kcal/mol/HA
Fit Quality
-5.95
FQ (Leeson)
HAC
37
heavy atoms
MW
505
Da
LogP
2.13
cLogP
Strain ΔE
33.7 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 33.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 10 Severe clashes 0
Final rank56.21558111624506Score-21.5097
Inter norm-0.581631Intra norm0.00028788
Top1000noExcludedno
Contacts18H-bonds1
Artifact reasongeometry warning; 18 clashes; 10 protein contact clashes
ResiduesA:ARG48;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR54;A:THR83;A:TRP47;A:VAL156;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.58RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
989 5.261315824560532 -0.603714 -16.1038 1 17 17 0.85 0.20 - no Open
986 5.770786952505254 -0.684306 -25.006 2 17 13 0.65 0.20 - no Open
982 6.831590296114315 -0.631332 -18.448 4 18 16 0.80 0.60 - no Open
999 8.21488777819133 -0.691017 -24.8564 2 20 14 0.70 0.20 - no Open
991 56.21558111624506 -0.581631 -21.5097 1 18 14 0.70 0.00 - no Current
983 56.846023674689064 -0.638341 -15.8179 5 19 15 0.75 0.20 - no Open
985 56.90596655947617 -0.616499 -22.3388 1 20 16 0.80 0.00 - no Open
992 57.12859200363561 -0.667155 -17.3578 2 17 14 0.70 0.20 - no Open
984 57.270324363866195 -0.650453 -21.9053 1 18 15 0.75 0.00 - no Open
1003 6.600791438983622 -0.600972 -24.8567 1 18 13 0.65 0.20 - yes Open
998 6.9864891900382 -0.591297 -19.3211 4 20 17 0.85 0.40 - yes Open
1004 56.51092702391629 -0.655942 -12.1454 2 14 14 0.70 0.20 - yes Open
997 57.303856470185664 -0.62455 -14.3072 4 18 17 0.85 0.60 - yes Open
993 57.37627785960962 -0.636806 -17.6957 0 19 16 0.80 0.00 - yes Open
987 57.53904655944858 -0.633541 -17.3119 1 13 10 0.50 0.00 - yes Open
990 57.69257254357571 -0.680225 -21.6112 3 20 16 0.80 0.40 - yes Open
996 57.96121863548281 -0.642077 -23.7322 2 14 13 0.65 0.20 - yes Open
994 58.22001385851653 -0.678188 -12.7809 1 21 17 0.85 0.20 - yes Open
981 59.37981478411859 -0.677603 -16.5586 2 19 17 0.85 0.00 - yes Open
1001 59.40316350507955 -0.636404 -18.9482 1 20 16 0.80 0.20 - yes Open
988 59.95131573285785 -0.613441 -16.5014 1 21 16 0.80 0.20 - yes Open
1000 60.513634966021684 -0.684577 -24.4245 2 18 12 0.60 0.20 - yes Open
995 62.1130761271655 -0.642347 -15.1306 1 20 17 0.85 0.20 - yes Open
1002 62.79162620982332 -0.748739 -22.3876 1 20 16 0.80 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.510kcal/mol
Ligand efficiency (LE) -0.5813kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -5.952
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 504.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.13
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 33.70kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 121.37kcal/mol
Minimised FF energy 87.67kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.