FAIRMol

OSA_Lib_1

Pose ID 42721 Compound 2659 Pose 634

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.438 kcal/mol/HA) ✓ Good fit quality (FQ -4.48) ✗ Very high strain energy (21.9 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-16.196
kcal/mol
LE
-0.438
kcal/mol/HA
Fit Quality
-4.48
FQ (Leeson)
HAC
37
heavy atoms
MW
535
Da
LogP
6.78
cLogP
Strain ΔE
21.9 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 5 Severe clashes 0
Final rank5.08809700459824Score-16.1959
Inter norm-0.527025Intra norm0.0892994
Top1000noExcludedno
Contacts14H-bonds1
Artifact reasongeometry warning; 17 clashes; 5 protein contact clashes; high strain Δ 20.8
ResiduesA:ASN22;A:CYS52;A:GLU18;A:GLY13;A:GLY49;A:ILE339;A:LEU17;A:MET113;A:SER109;A:SER14;A:THR335;A:TRP21;A:TYR110;A:VAL53

Protein summary

493 residues
Protein targetT18Atoms7550
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts13
PoseOpen native poseH-bonds0
IFP residuesA:ASP116; A:GLU18; A:GLY112; A:ILE106; A:LEU17; A:MET113; A:SER109; A:THR117; A:THR335; A:TRP21; A:TYR110; A:VAL53; A:VAL58
Current overlap8Native recall0.62
Jaccard0.42RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
716 4.696849092801991 -0.669437 -20.4248 0 18 0 0.00 - - no Open
720 4.859626902168574 -0.652673 -21.7584 0 18 0 0.00 - - no Open
730 4.909651590978486 -0.617771 -18.9521 1 17 0 0.00 - - no Open
722 4.973597256723719 -0.516772 -19.0104 1 14 0 0.00 - - no Open
631 4.996733076053392 -0.488834 -14.8783 0 12 10 0.77 - - no Open
634 5.08809700459824 -0.527025 -16.1959 1 14 8 0.62 - - no Current
733 5.150248905347559 -0.551923 -19.8858 1 16 0 0.00 - - no Open
630 5.169980110018646 -0.52551 -18.2584 1 14 8 0.62 - - no Open
723 5.188706576946113 -0.54103 -17.073 1 14 0 0.00 - - no Open
717 5.409238992016449 -0.501638 -17.3718 0 14 0 0.00 - - no Open
728 5.95663915500904 -0.671792 -21.805 0 18 0 0.00 - - no Open
632 54.7436311084979 -0.392619 -10.8663 0 9 9 0.69 - - no Open
633 54.97047852034492 -0.405526 -14.1493 0 9 9 0.69 - - no Open
635 55.06922744403984 -0.550582 -17.33 1 14 8 0.62 - - no Open
628 55.497981154103485 -0.468398 -14.5055 1 12 10 0.77 - - no Open
721 55.533799599150264 -0.579056 -16.5165 2 18 0 0.00 - - no Open
725 55.60668041830055 -0.582545 -20.1038 2 14 0 0.00 - - no Open
719 55.761676815425815 -0.59739 -18.7823 0 19 0 0.00 - - no Open
731 56.35264012966993 -0.638173 -21.7217 1 16 0 0.00 - - no Open
734 56.680506561019705 -0.619632 -18.5334 1 16 0 0.00 - - no Open
727 56.76921668168278 -0.595547 -18.3942 0 19 0 0.00 - - no Open
718 7.727185877664056 -0.535375 -16.6568 1 16 0 0.00 - - yes Open
629 56.08431882237537 -0.490886 -17.4451 0 10 10 0.77 - - yes Open
724 56.767821516922034 -0.511431 -17.33 0 14 0 0.00 - - yes Open
732 57.176581128438094 -0.540345 -18.6848 0 15 0 0.00 - - yes Open
729 57.625484230446006 -0.573041 -20.1712 0 16 0 0.00 - - yes Open
726 58.603996604781145 -0.563408 -15.4712 1 19 0 0.00 - - yes Open
715 60.01498287678175 -0.594937 -18.969 0 17 0 0.00 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -16.196kcal/mol
Ligand efficiency (LE) -0.4377kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.481
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 534.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 6.78
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 21.94kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 114.42kcal/mol
Minimised FF energy 92.48kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.