FAIRMol

OSA_Lib_70

Pose ID 4271 Compound 495 Pose 953

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.649 kcal/mol/HA) ✓ Good fit quality (FQ -6.38) ✗ Very high strain energy (27.4 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-20.760
kcal/mol
LE
-0.649
kcal/mol/HA
Fit Quality
-6.38
FQ (Leeson)
HAC
32
heavy atoms
MW
475
Da
LogP
3.78
cLogP
Strain ΔE
27.4 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 27.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 13 Severe clashes 2
Final rank58.67929402755901Score-20.7597
Inter norm-0.781213Intra norm0.132472
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 15 clashes; 2 protein clashes
ResiduesA:ALA32;A:ASP52;A:GLU43;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR180;A:THR83;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.77RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
911 3.28212585080371 -0.464422 -14.556 2 11 0 0.00 0.00 - no Open
955 3.41986828203709 -0.775874 -24.2002 0 20 17 0.85 0.00 - no Open
910 3.7811810184138266 -0.465799 -14.5043 2 10 0 0.00 0.00 - no Open
746 3.9092122471539077 -0.528601 -14.6552 1 11 0 0.00 0.00 - no Open
909 3.913689556569143 -0.551457 -18.5656 1 13 0 0.00 0.00 - no Open
744 4.391479998870725 -0.650554 -18.1005 2 9 0 0.00 0.00 - no Open
1103 4.539778637786404 -0.707267 -21.9306 2 15 0 0.00 0.00 - no Open
747 5.2426007962111365 -0.537275 -12.5725 2 8 0 0.00 0.00 - no Open
956 5.315681713377635 -0.849662 -25.4041 0 20 16 0.80 0.00 - no Open
1101 5.633438956740092 -0.737804 -21.8692 3 14 1 0.05 0.00 - no Open
1104 6.073538714598687 -0.696198 -17.2604 3 15 1 0.05 0.00 - no Open
912 54.93484532902622 -0.4982 -14.0944 2 11 0 0.00 0.00 - no Open
1102 55.204244254502605 -0.767597 -22.8323 2 17 1 0.05 0.00 - no Open
954 7.458471852044997 -0.75739 -18.7466 0 19 16 0.80 0.00 - yes Open
745 55.40874057995131 -0.495628 -14.8019 2 9 0 0.00 0.00 - yes Open
953 58.67929402755901 -0.781213 -20.7597 1 19 17 0.85 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.760kcal/mol
Ligand efficiency (LE) -0.6487kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.380
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 474.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.78
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 27.42kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 160.44kcal/mol
Minimised FF energy 133.03kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.