FAIRMol

OSA_Lib_50

Pose ID 4157 Compound 662 Pose 839

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.601 kcal/mol/HA) ✓ Good fit quality (FQ -6.15) ✗ Very high strain energy (37.2 kcal/mol) ✗ No H-bonds detected ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-22.237
kcal/mol
LE
-0.601
kcal/mol/HA
Fit Quality
-6.15
FQ (Leeson)
HAC
37
heavy atoms
MW
503
Da
LogP
1.49
cLogP
Strain ΔE
37.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 37.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 0 Hydrophobic 24 π–π 0 Clashes 6 Severe clashes 0
Final rank6.278877418186959Score-22.2368
Inter norm-0.630413Intra norm0.0294172
Top1000noExcludedno
Contacts21H-bonds0
Artifact reasongeometry warning; 16 clashes; 6 protein contact clashes; high strain Δ 38.3
ResiduesA:ALA32;A:ARG48;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:SER44;A:SER86;A:THR54;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.64RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

No hydrogen bonds detected for this pose.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
838 5.746295082926722 -0.633659 -23.7415 1 18 14 0.70 0.00 - no Open
846 6.228836469128684 -0.665054 -22.3963 1 21 17 0.85 0.00 - no Open
839 6.278877418186959 -0.630413 -22.2368 0 21 16 0.80 0.00 - no Current
837 54.50402717537393 -0.61119 -23.4132 1 20 16 0.80 0.00 - no Open
845 55.39038238999504 -0.668459 -27.5837 1 19 15 0.75 0.00 - no Open
835 55.58333334181339 -0.67306 -24.6555 2 19 18 0.90 0.00 - no Open
848 55.60494141037207 -0.65039 -22.9969 1 16 14 0.70 0.00 - no Open
833 55.79342338456338 -0.660432 -24.3608 0 15 11 0.55 0.00 - no Open
841 55.885010971957115 -0.582837 -22.3624 2 19 15 0.75 0.00 - no Open
844 56.21962285007319 -0.666799 -22.8698 1 16 14 0.70 0.00 - no Open
842 57.14577171923913 -0.61889 -22.7723 1 18 16 0.80 0.00 - yes Open
834 57.18630119595892 -0.605467 -27.3099 1 14 11 0.55 0.00 - yes Open
840 58.14268712580174 -0.62168 -21.774 0 21 16 0.80 0.00 - yes Open
847 59.013361746090695 -0.679696 -24.0484 2 13 10 0.50 0.20 - yes Open
836 59.589240734367785 -0.572322 -24.6522 1 14 12 0.60 0.00 - yes Open
843 60.850392885450226 -0.603725 -15.3959 1 20 16 0.80 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.237kcal/mol
Ligand efficiency (LE) -0.6010kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.153
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 502.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.49
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 37.18kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 215.78kcal/mol
Minimised FF energy 178.60kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.