FAIRMol

OSA_Lib_43

Pose ID 4143 Compound 642 Pose 825

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.602 kcal/mol/HA) ✓ Good fit quality (FQ -6.12) ✓ Good H-bonds (4 bonds) ✗ Very high strain energy (36.0 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.662
kcal/mol
LE
-0.602
kcal/mol/HA
Fit Quality
-6.12
FQ (Leeson)
HAC
36
heavy atoms
MW
490
Da
LogP
3.15
cLogP
Strain ΔE
36.0 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 36.0 kcal/mol

Interaction summary

Collapsible panels
H-bonds 4 Hydrophobic 24 π–π 2 Clashes 14 Severe clashes 2
Final rank59.93161040595322Score-21.6618
Inter norm-0.700894Intra norm0.0991765
Top1000noExcludedyes
Contacts21H-bonds4
Artifact reasonexcluded; geometry warning; 20 clashes; 2 protein clashes
ResiduesA:ALA32;A:ARG48;A:ASP52;A:CYS155;A:GLY157;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:TRP47;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap15Native recall0.75
Jaccard0.58RMSD-
H-bond strict3Strict recall0.43
H-bond same residue+role3Role recall0.60
H-bond same residue3Residue recall0.60

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
725 5.199885171737721 -0.373154 -11.7603 2 15 0 0.00 0.00 - no Open
813 5.438724231327866 -0.613242 -17.8402 1 17 13 0.65 0.20 - no Open
723 5.695403228454068 -0.48202 -11.8762 5 10 0 0.00 0.00 - no Open
618 5.779813374236834 -0.507317 -17.5796 3 13 0 0.00 0.00 - no Open
628 5.88661790051481 -0.445314 -15.2601 1 12 0 0.00 0.00 - no Open
810 6.071782156386927 -0.635258 -16.9639 3 17 16 0.80 0.60 - no Open
817 6.138229816692879 -0.603963 -13.4544 1 17 17 0.85 0.20 - no Open
829 6.188492676857888 -0.692845 -24.9088 2 19 17 0.85 0.00 - no Open
832 6.3110502613069 -0.610485 -21.7531 2 15 13 0.65 0.20 - no Open
721 6.510682654594804 -0.374439 -14.4296 2 14 0 0.00 0.00 - no Open
620 6.76614321635318 -0.408022 -12.4639 3 12 0 0.00 0.00 - no Open
824 55.03577249093066 -0.656758 -22.8915 1 15 13 0.65 0.00 - no Open
814 55.27974486958857 -0.705705 -24.2204 2 17 13 0.65 0.20 - no Open
822 55.358303497511955 -0.709666 -22.4297 3 18 14 0.70 0.20 - no Open
615 55.387057998275594 -0.458053 -12.8361 2 12 0 0.00 0.00 - no Open
816 55.39732143466571 -0.601715 -14.7845 2 14 13 0.65 0.00 - no Open
823 56.245860078715694 -0.643961 -22.6062 2 16 13 0.65 0.20 - no Open
827 6.753989161066888 -0.763512 -27.1071 4 20 18 0.90 0.60 - yes Open
732 55.509814002780686 -0.445583 -15.1562 4 12 0 0.00 0.00 - yes Open
815 55.8151728838121 -0.666318 -24.5877 2 17 13 0.65 0.20 - yes Open
726 55.82624142422725 -0.544834 -17.1273 5 16 0 0.00 0.00 - yes Open
809 55.884853218744134 -0.712385 -21.9714 3 18 17 0.85 0.60 - yes Open
821 55.91760706468468 -0.688925 -18.6027 2 18 14 0.70 0.20 - yes Open
735 56.033940821903826 -0.512937 -16.6195 2 12 0 0.00 0.00 - yes Open
736 56.15690983372645 -0.531885 -15.6928 4 11 0 0.00 0.00 - yes Open
811 56.272050947894876 -0.703589 -14.4132 4 18 16 0.80 0.60 - yes Open
727 56.57152165724404 -0.495203 -16.4483 4 15 0 0.00 0.00 - yes Open
730 56.63752702801069 -0.461127 -12.0861 3 11 0 0.00 0.00 - yes Open
626 56.687903728124695 -0.578336 -10.0774 2 16 0 0.00 0.00 - yes Open
831 56.72188223439526 -0.617275 -7.48477 1 16 15 0.75 0.20 - yes Open
617 57.039624301924675 -0.492991 -18.7104 1 14 0 0.00 0.00 - yes Open
830 57.158894875502995 -0.686879 -23.4326 5 18 15 0.75 0.60 - yes Open
627 57.17316114486377 -0.495594 -14.5016 3 12 0 0.00 0.00 - yes Open
629 57.18042319281949 -0.52033 -19.2153 6 12 0 0.00 0.00 - yes Open
731 57.314009543389886 -0.519995 -16.3468 3 12 0 0.00 0.00 - yes Open
722 57.37494547872849 -0.469582 -16.0651 2 17 0 0.00 0.00 - yes Open
826 57.5399059241514 -0.73814 -13.1352 4 19 15 0.75 0.60 - yes Open
625 57.623684632372495 -0.529004 -13.5881 1 13 0 0.00 0.00 - yes Open
820 57.63629711858755 -0.659707 -20.6912 0 15 13 0.65 0.00 - yes Open
624 57.73854054201422 -0.585526 -19.5347 7 10 0 0.00 0.00 - yes Open
728 57.7928563403071 -0.50665 -15.4666 3 14 0 0.00 0.00 - yes Open
818 57.825021263165006 -0.63386 -16.1063 2 13 10 0.50 0.00 - yes Open
724 58.042435412022456 -0.438091 -10.5396 3 11 0 0.00 0.00 - yes Open
729 58.191732226554755 -0.440114 -9.83591 3 10 0 0.00 0.00 - yes Open
819 58.30916741085935 -0.703206 -19.838 1 20 16 0.80 0.20 - yes Open
622 58.58757294992907 -0.508848 -16.5846 3 12 0 0.00 0.00 - yes Open
616 58.66803904314661 -0.701244 -14.3967 4 12 0 0.00 0.00 - yes Open
733 59.002846100583334 -0.563769 -16.8478 4 13 0 0.00 0.00 - yes Open
734 59.460376526810194 -0.537622 -16.7143 4 13 0 0.00 0.00 - yes Open
623 59.58379506226615 -0.52905 -17.777 3 12 0 0.00 0.00 - yes Open
828 59.88941444782486 -0.633467 -18.4391 2 18 16 0.80 0.00 - yes Open
825 59.93161040595322 -0.700894 -21.6618 4 21 15 0.75 0.60 - yes Current
812 60.27085877012976 -0.67077 -23.4406 2 19 16 0.80 0.00 - yes Open
619 60.63469808226914 -0.519981 -18.5032 3 12 0 0.00 0.00 - yes Open
614 60.72631531866858 -0.529667 -15.7272 3 13 0 0.00 0.00 - yes Open
621 61.435183854339286 -0.491928 -12.9227 5 13 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.662kcal/mol
Ligand efficiency (LE) -0.6017kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.116
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 36HA

Physicochemical properties

Molecular weight 489.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.15
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 35.95kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 110.10kcal/mol
Minimised FF energy 74.15kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.