FAIRMol

OSA_Lib_23

Pose ID 4097 Compound 561 Pose 779

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.824 kcal/mol/HA) ✓ Good fit quality (FQ -8.11) ✗ Very high strain energy (22.9 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-26.372
kcal/mol
LE
-0.824
kcal/mol/HA
Fit Quality
-8.11
FQ (Leeson)
HAC
32
heavy atoms
MW
476
Da
LogP
3.11
cLogP
Strain ΔE
22.9 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 22.9 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 10 Severe clashes 2
Final rank57.2261228474444Score-26.3724
Inter norm-0.893563Intra norm0.0694254
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 13 clashes; 2 protein clashes
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:TRP47;A:TYR162;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap15Native recall0.75
Jaccard0.62RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
784 4.340418524383093 -0.757525 -23.7416 1 19 16 0.80 0.20 - no Open
748 4.789405360951812 -0.685116 -21.5465 3 16 1 0.05 0.00 - no Open
778 4.802068615670731 -0.67629 -19.7901 0 18 15 0.75 0.00 - no Open
742 4.985372977299745 -0.8543 -24.7081 4 15 1 0.05 0.00 - no Open
775 5.031294907009333 -0.696668 -20.9918 0 16 15 0.75 0.00 - no Open
783 5.165149154441218 -0.645272 -19.3358 0 17 15 0.75 0.00 - no Open
777 5.283295736017563 -0.766078 -25.5034 0 17 15 0.75 0.00 - no Open
749 5.315861828592169 -0.679466 -19.4014 3 15 1 0.05 0.00 - no Open
741 5.693979193643358 -0.748364 -21.8242 4 13 0 0.00 0.00 - no Open
740 6.386496695805026 -0.614226 -17.8216 3 14 1 0.05 0.00 - no Open
754 7.047674852930161 -0.681204 -19.5325 3 15 1 0.05 0.00 - no Open
776 54.19192495738549 -0.792625 -22.7459 0 19 16 0.80 0.00 - no Open
752 5.787850833341128 -0.614926 -18.7937 3 14 1 0.05 0.00 - yes Open
747 6.251409771195268 -0.624602 -18.1682 2 12 0 0.00 0.00 - yes Open
785 6.925103903821261 -0.803088 -25.2179 1 19 16 0.80 0.00 - yes Open
753 8.14130536068911 -0.735296 -19.714 4 11 0 0.00 0.00 - yes Open
774 55.02279697118261 -0.677019 -20.5339 0 16 15 0.75 0.00 - yes Open
743 55.36444697198205 -0.612662 -19.8329 3 16 1 0.05 0.00 - yes Open
787 55.87287724411718 -0.806721 -24.5189 1 20 16 0.80 0.00 - yes Open
788 56.068594449744154 -0.856492 -22.4408 1 18 14 0.70 0.00 - yes Open
782 56.10230779739426 -0.711074 -21.931 0 16 15 0.75 0.00 - yes Open
750 56.212337480928284 -0.588608 -18.583 3 15 1 0.05 0.00 - yes Open
757 56.898512794378306 -0.665433 -20.944 2 12 0 0.00 0.00 - yes Open
746 56.9735987506083 -0.731742 -22.0924 5 14 1 0.05 0.00 - yes Open
786 57.020530183666594 -0.661697 -19.8078 1 17 15 0.75 0.20 - yes Open
779 57.2261228474444 -0.893563 -26.3724 1 19 15 0.75 0.00 - yes Current
755 57.36065100177839 -0.657894 -21.2804 4 14 1 0.05 0.00 - yes Open
780 57.4082283679076 -0.91664 -25.029 2 18 14 0.70 0.00 - yes Open
758 57.45166151440917 -0.678024 -18.4681 3 12 1 0.05 0.00 - yes Open
773 57.52288062100218 -0.640738 -16.106 1 17 16 0.80 0.20 - yes Open
751 57.730046600408926 -0.590373 -18.4773 1 18 1 0.05 0.00 - yes Open
745 57.92997605201672 -0.794459 -21.7516 5 14 1 0.05 0.00 - yes Open
744 58.39868436337761 -0.775625 -19.6978 4 17 1 0.05 0.00 - yes Open
781 58.868358854299814 -0.658566 -21.7467 0 17 15 0.75 0.00 - yes Open
756 59.742434966387954 -0.755555 -19.2954 5 16 1 0.05 0.00 - yes Open
739 60.43758286928337 -0.627951 -17.7115 5 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -26.372kcal/mol
Ligand efficiency (LE) -0.8241kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -8.105
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 475.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.11
Lipinski: ≤ 5
Rotatable bonds 5

Conformational strain (MMFF94s)

Strain energy (ΔE) 22.92kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 155.25kcal/mol
Minimised FF energy 132.33kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.