FAIRMol

OSA_Lib_21

Pose ID 4080 Compound 566 Pose 762

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.614 kcal/mol/HA) ✓ Good fit quality (FQ -6.28) ✗ Very high strain energy (26.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-22.708
kcal/mol
LE
-0.614
kcal/mol/HA
Fit Quality
-6.28
FQ (Leeson)
HAC
37
heavy atoms
MW
503
Da
LogP
1.49
cLogP
Strain ΔE
26.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 26.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 2 Clashes 8 Severe clashes 1
Final rank56.809215515860934Score-22.7082
Inter norm-0.697034Intra norm0.0832985
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 17 clashes; 1 protein clash
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:SER86;A:THR54;A:THR83;A:TRP47;A:TYR162;A:VAL30;A:VAL31;A:VAL49;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.70RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
648 3.654048777040276 -0.460593 -18.7111 1 10 0 0.00 0.00 - no Open
650 4.276327406338073 -0.473844 -18.113 1 10 0 0.00 0.00 - no Open
757 4.470783622620282 -0.564526 -18.871 2 18 13 0.65 0.00 - no Open
652 4.988962342108749 -0.456595 -16.3848 2 11 0 0.00 0.00 - no Open
749 5.007481566539756 -0.568231 -18.2276 0 18 13 0.65 0.00 - no Open
759 5.1902556663508 -0.617813 -21.2356 1 19 14 0.70 0.20 - no Open
640 5.204641784337701 -0.412403 -11.0914 2 10 0 0.00 0.00 - no Open
751 5.232239438700562 -0.606627 -19.6771 0 18 13 0.65 0.00 - no Open
771 5.28324080082365 -0.573935 -18.3575 0 14 10 0.50 0.00 - no Open
642 5.913373748990659 -0.396204 -14.8692 2 9 0 0.00 0.00 - no Open
758 6.310439773447799 -0.56831 -19.2357 1 16 14 0.70 0.00 - no Open
644 6.607181796605833 -0.404749 -12.5783 1 10 0 0.00 0.00 - no Open
768 7.0583281576802 -0.634418 -22.0687 1 17 15 0.75 0.00 - no Open
772 7.154793813516009 -0.551023 -15.4795 0 13 9 0.45 0.00 - no Open
753 7.641119035703079 -0.580197 -22.5272 1 17 13 0.65 0.00 - no Open
654 53.67795360127522 -0.45806 -13.4492 2 9 0 0.00 0.00 - no Open
647 54.42781281342558 -0.407712 -12.8784 1 11 0 0.00 0.00 - no Open
655 54.557847021330616 -0.380001 -12.5835 1 11 0 0.00 0.00 - no Open
752 56.11766390368315 -0.689924 -24.4634 1 19 16 0.80 0.00 - no Open
763 56.14896048770573 -0.670928 -24.0801 1 15 11 0.55 0.00 - no Open
750 56.261934033309416 -0.608479 -18.4468 0 21 16 0.80 0.00 - no Open
760 56.33449369464164 -0.660562 -22.1644 1 17 15 0.75 0.00 - no Open
646 55.35347237282498 -0.382487 -14.0081 1 9 0 0.00 0.00 - yes Open
645 55.40229001611615 -0.534679 -18.8382 3 14 0 0.00 0.00 - yes Open
761 55.51051473398724 -0.650436 -19.1027 0 17 15 0.75 0.00 - yes Open
643 55.699087167352815 -0.463505 -17.4386 3 13 0 0.00 0.00 - yes Open
765 55.75691810755007 -0.61185 -21.5002 1 18 15 0.75 0.20 - yes Open
653 55.83419170326622 -0.376397 -13.1292 4 10 0 0.00 0.00 - yes Open
764 56.331713135523 -0.578755 -17.3039 0 14 11 0.55 0.00 - yes Open
769 56.39287016389826 -0.580772 -22.3616 1 15 11 0.55 0.00 - yes Open
641 56.42794222808606 -0.471519 -14.9788 3 11 0 0.00 0.00 - yes Open
770 56.6372303362315 -0.686759 -20.6889 0 21 17 0.85 0.00 - yes Open
649 56.67979554622855 -0.467635 -17.6656 3 12 0 0.00 0.00 - yes Open
767 56.74191448450843 -0.700959 -18.0036 2 20 17 0.85 0.40 - yes Open
762 56.809215515860934 -0.697034 -22.7082 1 19 16 0.80 0.00 - yes Current
755 57.40935423509804 -0.697033 -22.5037 2 19 16 0.80 0.20 - yes Open
766 57.48102088371495 -0.620407 -21.2466 1 17 13 0.65 0.20 - yes Open
756 57.52316110628624 -0.635409 -19.8797 2 17 17 0.85 0.20 - yes Open
754 58.23659201973931 -0.672207 -19.8644 0 20 17 0.85 0.00 - yes Open
651 59.161335702096714 -0.563468 -19.4954 2 16 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -22.708kcal/mol
Ligand efficiency (LE) -0.6137kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.283
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 502.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) 1.49
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 26.12kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 157.67kcal/mol
Minimised FF energy 131.55kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.