FAIRMol

OSA_Lib_1

Pose ID 3990 Compound 538 Pose 672

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.659 kcal/mol/HA) ✓ Good fit quality (FQ -6.75) ✗ Very high strain energy (23.2 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-24.387
kcal/mol
LE
-0.659
kcal/mol/HA
Fit Quality
-6.75
FQ (Leeson)
HAC
37
heavy atoms
MW
535
Da
LogP
6.78
cLogP
Strain ΔE
23.2 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 23.2 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 11 Severe clashes 0
Final rank6.747198210916205Score-24.3875
Inter norm-0.638524Intra norm-0.0205975
Top1000noExcludedno
Contacts14H-bonds1
Artifact reasongeometry warning; 17 clashes; 11 protein contact clashes; high strain Δ 20.5
ResiduesA:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:PHE56;A:PHE91;A:PRO50;A:PRO88;A:SER86;A:THR54;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap12Native recall0.60
Jaccard0.55RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
661 3.9534125250212915 -0.539084 -17.6713 0 16 15 0.75 0.00 - no Open
670 5.302911838111157 -0.623143 -20.7284 0 13 12 0.60 0.00 - no Open
673 5.376951321364157 -0.721597 -20.3615 0 21 17 0.85 0.00 - no Open
665 5.602785480619648 -0.58204 -17.5327 0 20 17 0.85 0.00 - no Open
662 6.204550274643658 -0.526159 -19.6742 0 18 15 0.75 0.00 - no Open
672 6.747198210916205 -0.638524 -24.3875 1 14 12 0.60 0.00 - no Current
671 56.705449159521564 -0.617882 -18.4392 0 17 14 0.70 0.00 - no Open
667 56.267585914789 -0.717017 -25.7859 0 19 15 0.75 0.00 - yes Open
675 56.65139428764116 -0.73125 -24.359 0 20 16 0.80 0.00 - yes Open
668 56.97328320901291 -0.676711 -19.4543 1 19 14 0.70 0.00 - yes Open
674 57.786442039934336 -0.636941 -22.9389 0 15 13 0.65 0.00 - yes Open
666 57.97573970045298 -0.636916 -19.4259 1 19 15 0.75 0.00 - yes Open
676 58.10712127191333 -0.631477 -19.497 0 17 14 0.70 0.00 - yes Open
664 58.44254164882153 -0.616315 -18.2137 1 21 16 0.80 0.00 - yes Open
669 58.48977165206177 -0.56872 -13.6682 0 14 11 0.55 0.00 - yes Open
663 59.19434258309486 -0.639883 -18.0876 1 20 16 0.80 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -24.387kcal/mol
Ligand efficiency (LE) -0.6591kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.748
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 534.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 6.78
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 23.25kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 115.00kcal/mol
Minimised FF energy 91.76kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.