FAIRMol

OHD_TbNat_130

Pose ID 389 Compound 453 Pose 389

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Good H-bonds (5 bonds) ✗ Very high strain energy (70.7 kcal/mol) ✗ Poor LE (-0.049 kcal/mol/HA) ✗ Geometry warnings ℹ SASA not computed
Score
-2.544
kcal/mol
LE
-0.049
kcal/mol/HA
Fit Quality
-0.54
FQ (Leeson)
HAC
52
heavy atoms
MW
737
Da
LogP
-0.86
cLogP
Strain ΔE
70.7 kcal/mol
SASA buried
computing…
Overall: Likely artefact or unreliable pose
Binding evidence: weak
Native-like contacts: strong
Ligand efficiency: weak
Geometry reliability: low
Reason: geometry warning, clashes, strain 70.7 kcal/mol

Interaction summary

Collapsible panels
H-bonds 5 Hydrophobic 24 π–π 1 Clashes 14 Severe clashes 3
Final rank62.42813676895114Score-2.54394
Inter norm-0.4332Intra norm0.384278
Top1000noExcludedyes
Contacts23H-bonds5
Artifact reasonexcluded; hard geometry fail; 1 severe clash; 3 protein clashes; high raw intra
ResiduesA:ALA10;A:ARG29;A:ARG71;A:ASN65;A:ASP22;A:GLN36;A:GLU31;A:GLY21;A:ILE61;A:ILE8;A:LEU23;A:LEU28;A:LEU68;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap19Native recall0.90
Jaccard0.76RMSD-
H-bond strict2Strict recall0.40
H-bond same residue+role2Role recall0.40
H-bond same residue2Residue recall0.40

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
381 10.373499739274774 -0.385665 -18.848 6 20 17 0.81 0.80 - no Open
385 11.983850414986405 -0.353816 -15.8876 6 17 13 0.62 0.20 - yes Open
382 13.093649115005693 -0.419965 -19.104 5 19 15 0.71 0.40 - yes Open
387 59.345346051523876 -0.497227 -9.64966 5 20 17 0.81 0.60 - yes Open
379 59.379527286450575 -0.475393 -15.0949 5 21 15 0.71 0.20 - yes Open
384 59.49001355012986 -0.432556 -15.2608 8 17 13 0.62 0.00 - yes Open
380 59.49075806035832 -0.373854 -5.47768 2 19 14 0.67 0.20 - yes Open
383 59.54674921664915 -0.48123 -9.05507 9 20 17 0.81 0.80 - yes Open
386 59.98347504726175 -0.413172 -7.4053 4 16 12 0.57 0.00 - yes Open
389 62.42813676895114 -0.4332 -2.54394 5 23 19 0.90 0.40 - yes Current
390 63.543063595624176 -0.360442 -0.568547 3 16 13 0.62 0.20 - yes Open
378 63.630196745953086 -0.477671 -22.5646 12 23 19 0.90 0.60 - yes Open
388 70.62242913881107 -0.411984 1.01744 8 21 16 0.76 0.60 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -2.544kcal/mol
Ligand efficiency (LE) -0.0489kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -0.542
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 52HA

Physicochemical properties

Molecular weight 736.8Da
Lipinski: ≤ 500 Da
LogP (cLogP) -0.86
Lipinski: ≤ 5
Rotatable bonds 8

Conformational strain (MMFF94s)

Strain energy (ΔE) 70.68kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 148.99kcal/mol
Minimised FF energy 78.31kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.