FAIRMol

KB_Leish_188

Pose ID 3897 Compound 699 Pose 579

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.594 kcal/mol/HA) ✓ Good fit quality (FQ -6.08) ✗ Very high strain energy (43.5 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-21.974
kcal/mol
LE
-0.594
kcal/mol/HA
Fit Quality
-6.08
FQ (Leeson)
HAC
37
heavy atoms
MW
496
Da
LogP
3.01
cLogP
Strain ΔE
43.5 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 43.5 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 3 Clashes 9 Severe clashes 1
Final rank8.261263508834592Score-21.9743
Inter norm-0.708317Intra norm0.114401
Top1000noExcludedyes
Contacts19H-bonds1
Artifact reasonexcluded; geometry warning; 17 clashes; 1 protein clash; high strain Δ 31.8
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:PRO93;A:THR83;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap17Native recall0.85
Jaccard0.77RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
394 4.824031120225275 -0.559793 -17.9593 0 16 0 0.00 0.00 - no Open
393 4.8342966363052895 -0.874586 -28.7263 2 16 0 0.00 0.00 - no Open
401 5.544913036571565 -0.837917 -25.4211 2 14 0 0.00 0.00 - no Open
524 5.71545161130506 -0.531814 -22.122 2 12 0 0.00 0.00 - no Open
523 5.853583757572163 -0.475833 -14.4118 4 13 0 0.00 0.00 - no Open
400 5.991578804880139 -0.6343 -23.2541 0 16 0 0.00 0.00 - no Open
533 6.016219807250548 -0.503386 -16.6918 1 13 0 0.00 0.00 - no Open
530 6.271765321214856 -0.532132 -26.5306 2 12 0 0.00 0.00 - no Open
717 6.359048231967443 -0.366984 -12.9882 3 9 0 0.00 0.00 - no Open
720 6.454657660615654 -0.439902 -16.8067 5 13 0 0.00 0.00 - no Open
538 6.461885054046319 -0.485127 -22.026 3 13 0 0.00 0.00 - no Open
588 6.469183471884971 -0.642205 -21.2297 1 18 17 0.85 0.20 - no Open
582 6.557615301449495 -0.660037 -17.1485 0 19 18 0.90 0.00 - no Open
712 6.820650888681524 -0.391361 -14.3591 3 12 0 0.00 0.00 - no Open
527 7.163080623390221 -0.625227 -23.7366 4 13 0 0.00 0.00 - no Open
583 7.391532983625233 -0.715721 -21.8731 1 17 15 0.75 0.20 - no Open
537 7.6183813565571885 -0.587778 -19.2357 2 16 0 0.00 0.00 - no Open
713 7.769950286759409 -0.481214 -15.2582 3 10 0 0.00 0.00 - no Open
536 8.260915333543338 -0.552057 -24.578 1 13 0 0.00 0.00 - no Open
718 8.686843616583896 -0.450704 -19.2841 4 15 0 0.00 0.00 - no Open
395 6.732147949674597 -0.704644 -25.0006 0 16 0 0.00 0.00 - yes Open
531 7.074134258414574 -0.475045 -19.5657 1 15 0 0.00 0.00 - yes Open
529 7.461715263826837 -0.463645 -17.571 0 14 0 0.00 0.00 - yes Open
528 7.486579424380058 -0.511433 -21.3373 5 14 0 0.00 0.00 - yes Open
587 7.531982670403918 -0.586933 -20.6302 0 14 11 0.55 0.00 - yes Open
397 7.780685289612809 -0.639316 -26.3868 1 15 0 0.00 0.00 - yes Open
534 7.870906154971624 -0.549002 -23.6055 1 14 0 0.00 0.00 - yes Open
398 7.953263128225099 -0.8172 -28.1181 2 16 0 0.00 0.00 - yes Open
719 8.062327028852009 -0.470867 -13.935 3 10 0 0.00 0.00 - yes Open
396 8.068583176739661 -0.769401 -19.7046 0 15 0 0.00 0.00 - yes Open
711 8.236743801116575 -0.579801 -22.5862 5 14 0 0.00 0.00 - yes Open
579 8.261263508834592 -0.708317 -21.9743 1 19 17 0.85 0.00 - yes Current
585 8.383207669517338 -0.707315 -24.7732 0 19 18 0.90 0.00 - yes Open
716 8.552341082283359 -0.374775 -12.8459 3 11 0 0.00 0.00 - yes Open
581 8.603768764228624 -0.683635 -27.2741 1 21 18 0.90 0.00 - yes Open
526 8.830135839323713 -0.478375 -19.3293 2 15 0 0.00 0.00 - yes Open
540 9.305664535969818 -0.553463 -23.5298 5 15 0 0.00 0.00 - yes Open
402 9.672259340185855 -0.599865 -14.2895 1 16 0 0.00 0.00 - yes Open
580 10.447446779426922 -0.645172 -24.8712 3 10 7 0.35 0.20 - yes Open
584 10.720186707206247 -0.783426 -21.1736 1 18 15 0.75 0.20 - yes Open
399 56.65304746631722 -0.56375 -17.945 0 15 0 0.00 0.00 - yes Open
532 57.0975813531502 -0.584451 -23.4639 1 13 0 0.00 0.00 - yes Open
539 57.32768770998607 -0.461476 -15.804 2 18 0 0.00 0.00 - yes Open
715 57.421555140899216 -0.539862 -20.0272 6 11 0 0.00 0.00 - yes Open
714 57.73022582961767 -0.443412 -16.8325 3 10 0 0.00 0.00 - yes Open
525 58.73819404495769 -0.410954 -18.5926 4 17 0 0.00 0.00 - yes Open
586 59.099750611742564 -0.791936 -27.0296 1 20 17 0.85 0.20 - yes Open
535 59.36500216101931 -0.535377 -21.3038 3 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -21.974kcal/mol
Ligand efficiency (LE) -0.5939kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.080
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 495.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.01
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 43.48kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 122.84kcal/mol
Minimised FF energy 79.36kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.