FAIRMol

KB_Leish_175

Pose ID 3894 Compound 584 Pose 576

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.666 kcal/mol/HA) ✓ Good fit quality (FQ -6.43) ✗ High strain energy (18.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-19.984
kcal/mol
LE
-0.666
kcal/mol/HA
Fit Quality
-6.43
FQ (Leeson)
HAC
30
heavy atoms
MW
404
Da
LogP
2.84
cLogP
Strain ΔE
18.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 18.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 7 Severe clashes 0
Final rank4.693917173896296Score-19.9839
Inter norm-0.844218Intra norm0.178089
Top1000noExcludedno
Contacts19H-bonds2
Artifact reasongeometry warning; 13 clashes; 7 protein contact clashes; high strain Δ 20.7
ResiduesA:ALA32;A:ARG97;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:SER86;A:THR54;A:THR83;A:TYR162;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap18Native recall0.90
Jaccard0.86RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
530 3.2057635565037708 -0.749907 -21.1874 2 17 1 0.05 0.00 - no Open
457 3.315080628835318 -0.791061 -25.5014 6 15 1 0.05 0.00 - no Open
529 3.481902399795697 -0.83408 -24.8519 2 20 1 0.05 0.00 - no Open
455 4.140245303416389 -0.724352 -20.9449 6 15 1 0.05 0.00 - no Open
576 4.693917173896296 -0.844218 -19.9839 2 19 18 0.90 0.20 - no Current
456 4.781246866948247 -0.714375 -22.3378 3 16 0 0.00 0.00 - no Open
422 8.476253130545862 -0.785771 -17.9194 6 19 1 0.05 0.00 - no Open
575 5.6692435087881945 -0.6935 -20.9743 1 17 11 0.55 0.00 - yes Open
454 6.462338453067334 -0.729474 -18.6328 4 17 0 0.00 0.00 - yes Open
419 9.97971793295765 -0.743713 -19.041 2 20 1 0.05 0.00 - yes Open
421 12.658290186532163 -0.63083 -12.9809 1 20 1 0.05 0.00 - yes Open
420 13.216744066065624 -0.693652 -17.2077 6 18 1 0.05 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -19.984kcal/mol
Ligand efficiency (LE) -0.6661kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.426
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 30HA

Physicochemical properties

Molecular weight 403.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 2.84
Lipinski: ≤ 5
Rotatable bonds 7

Conformational strain (MMFF94s)

Strain energy (ΔE) 18.05kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -59.34kcal/mol
Minimised FF energy -77.39kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.