FAIRMol

KB_Leish_46

Pose ID 3863 Compound 574 Pose 545

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.749 kcal/mol/HA) ✓ Good fit quality (FQ -7.37) ✗ Very high strain energy (21.1 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-23.965
kcal/mol
LE
-0.749
kcal/mol/HA
Fit Quality
-7.37
FQ (Leeson)
HAC
32
heavy atoms
MW
478
Da
LogP
3.61
cLogP
Strain ΔE
21.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 21.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 24 π–π 1 Clashes 10 Severe clashes 2
Final rank56.76538553890124Score-23.9649
Inter norm-0.749641Intra norm0.00073844
Top1000noExcludedyes
Contacts20H-bonds1
Artifact reasonexcluded; geometry warning; 9 clashes; 2 protein clashes
ResiduesA:ALA32;A:ARG48;A:ASP52;A:ILE45;A:LEU94;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR180;A:TRP47;A:TYR162;A:TYR178;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap16Native recall0.80
Jaccard0.67RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role0Role recall0.00
H-bond same residue0Residue recall0.00

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
539 4.578051279948418 -0.836441 -23.7077 1 21 18 0.90 0.20 - no Open
531 4.873103504307923 -0.755991 -21.9113 1 21 18 0.90 0.20 - no Open
544 4.957947154718397 -0.77194 -27.5356 1 16 13 0.65 0.00 - no Open
424 4.9786679789210915 -0.607541 -14.4757 3 13 1 0.05 0.00 - no Open
547 5.35220158640997 -0.788979 -23.0974 2 19 17 0.85 0.20 - no Open
418 5.503663179548383 -0.591602 -15.7788 4 14 0 0.00 0.00 - no Open
536 5.592270017366477 -0.760386 -20.7067 1 16 14 0.70 0.00 - no Open
421 6.130453196567059 -0.634935 -20.8308 3 14 1 0.05 0.00 - no Open
416 55.392362047497045 -0.680698 -16.8839 5 13 1 0.05 0.00 - no Open
422 56.08470595499364 -0.652427 -20.7805 5 14 0 0.00 0.00 - no Open
532 5.351274929047857 -0.708091 -23.2492 1 17 16 0.80 0.00 - yes Open
428 54.92680923743816 -0.612277 -17.4971 2 12 0 0.00 0.00 - yes Open
542 54.93402315854781 -0.805458 -25.2612 1 18 16 0.80 0.00 - yes Open
543 55.11394031842511 -0.719767 -20.2266 1 15 13 0.65 0.00 - yes Open
538 55.320432949481805 -0.847022 -26.2041 1 17 16 0.80 0.00 - yes Open
554 55.44674008211802 -0.826456 -27.7497 1 17 16 0.80 0.00 - yes Open
425 55.634847078930164 -0.69617 -22.5042 4 16 0 0.00 0.00 - yes Open
426 55.978226159919124 -0.653399 -24.2595 3 15 0 0.00 0.00 - yes Open
419 56.099292180823014 -0.726868 -22.5368 5 16 0 0.00 0.00 - yes Open
550 56.15369218492761 -0.823781 -27.1051 2 15 12 0.60 0.00 - yes Open
417 56.17706705702731 -0.608003 -12.7259 4 15 1 0.05 0.00 - yes Open
549 56.491681708803526 -0.740201 -25.7463 3 10 9 0.45 0.20 - yes Open
541 56.59007578258512 -0.764635 -20.806 1 18 15 0.75 0.00 - yes Open
420 56.64458233008418 -0.722115 -24.8227 3 12 0 0.00 0.00 - yes Open
545 56.76538553890124 -0.749641 -23.9649 1 20 16 0.80 0.00 - yes Current
430 56.8614587127542 -0.587938 -18.1571 1 14 0 0.00 0.00 - yes Open
534 56.898701725433426 -0.808824 -25.7914 1 18 14 0.70 0.00 - yes Open
552 56.90385083398705 -0.809357 -17.8446 3 13 11 0.55 0.20 - yes Open
535 57.056440842723944 -0.775288 -21.1576 1 19 16 0.80 0.00 - yes Open
537 57.14621584789709 -0.765841 -16.9705 2 16 13 0.65 0.00 - yes Open
540 57.43980407676235 -0.676081 -18.3247 1 19 18 0.90 0.00 - yes Open
548 57.858147270023764 -0.720473 -17.1943 1 16 14 0.70 0.00 - yes Open
533 58.61620205238415 -0.770822 -25.5399 1 18 16 0.80 0.00 - yes Open
553 59.357423973642355 -0.702808 -22.5276 2 17 13 0.65 0.00 - yes Open
427 59.49085344586227 -0.705055 -24.2427 2 14 0 0.00 0.00 - yes Open
429 60.01765742426803 -0.678756 -20.4807 2 16 0 0.00 0.00 - yes Open
551 60.04628309910173 -0.822051 -24.2471 1 18 14 0.70 0.00 - yes Open
546 60.6066765495306 -0.925317 -25.6492 3 14 12 0.60 0.20 - yes Open
431 61.29124134893323 -0.652682 -23.0277 5 15 0 0.00 0.00 - yes Open
423 61.42540633024061 -0.656692 -19.582 4 15 1 0.05 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.965kcal/mol
Ligand efficiency (LE) -0.7489kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.365
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 32HA

Physicochemical properties

Molecular weight 478.4Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.61
Lipinski: ≤ 5
Rotatable bonds 4

Conformational strain (MMFF94s)

Strain energy (ΔE) 21.07kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 55.05kcal/mol
Minimised FF energy 33.98kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.