FAIRMol

KB_Leish_34

Pose ID 3825 Compound 153 Pose 507

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.765 kcal/mol/HA) ✓ Good fit quality (FQ -7.45) ✓ Strong H-bond network (7 bonds) ✗ Very high strain energy (39.3 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-23.712
kcal/mol
LE
-0.765
kcal/mol/HA
Fit Quality
-7.45
FQ (Leeson)
HAC
31
heavy atoms
MW
418
Da
LogP
3.00
cLogP
Strain ΔE
39.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 39.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 7 Hydrophobic 24 π–π 2 Clashes 11 Severe clashes 0
Final rank55.93854545562736Score-23.7117
Inter norm-0.927731Intra norm0.162837
Top1000noExcludedno
Contacts18H-bonds7
Artifact reasongeometry warning; 17 clashes; 11 protein contact clashes; high strain Δ 40.4
ResiduesA:ARG48;A:ARG97;A:GLU43;A:ILE45;A:LEU94;A:LYS57;A:LYS90;A:LYS95;A:MET53;A:NDP301;A:PHE56;A:PHE91;A:PRO46;A:PRO88;A:SER44;A:SER86;A:TRP47;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap11Native recall0.55
Jaccard0.41RMSD-
H-bond strict1Strict recall0.14
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
657 4.2704193353870785 -0.844612 -23.4937 5 17 0 0.00 0.00 - no Open
133 5.417368585019053 -0.937561 -26.8058 6 18 0 0.00 0.00 - no Open
134 5.4255427326367345 -0.991392 -29.475 5 19 0 0.00 0.00 - no Open
132 5.468686276653935 -1.00923 -30.0975 6 18 0 0.00 0.00 - no Open
508 6.063865071119024 -0.878702 -24.0407 10 19 15 0.75 0.80 - no Open
480 6.1076766813231425 -0.733522 -21.2295 2 15 1 0.05 0.00 - no Open
482 6.452309044329518 -0.784431 -21.6759 5 17 1 0.05 0.00 - no Open
479 7.339930842303011 -0.923564 -26.714 6 20 1 0.05 0.00 - no Open
507 55.93854545562736 -0.927731 -23.7117 7 18 11 0.55 0.20 - no Current
656 6.666237321815385 -0.761865 -23.841 7 21 0 0.00 0.00 - yes Open
510 7.202003981104733 -0.907111 -22.8871 6 20 16 0.80 0.80 - yes Open
509 8.645096920148294 -0.880769 -21.533 10 17 14 0.70 0.80 - yes Open
135 57.5490545506712 -0.912678 -25.1879 5 17 0 0.00 0.00 - yes Open
481 60.8641049522853 -0.78431 -20.1283 4 12 1 0.05 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -23.712kcal/mol
Ligand efficiency (LE) -0.7649kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.452
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 31HA

Physicochemical properties

Molecular weight 418.5Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.00
Lipinski: ≤ 5
Rotatable bonds 6

Conformational strain (MMFF94s)

Strain energy (ΔE) 39.31kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy -76.43kcal/mol
Minimised FF energy -115.73kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.