FAIRMol

OHD_TbNat_129

Pose ID 372 Compound 456 Pose 372

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✗ Very high strain energy (60.4 kcal/mol) ✗ Poor LE (0.130 kcal/mol/HA) ✗ Poor fit quality (FQ 1.47) ✗ Geometry warnings ℹ SASA not computed
Score
7.539
kcal/mol
LE
0.130
kcal/mol/HA
Fit Quality
1.47
FQ (Leeson)
HAC
58
heavy atoms
MW
823
Da
LogP
0.27
cLogP
Strain ΔE
60.4 kcal/mol
SASA buried
computing…
Overall: Likely artefact or unreliable pose
Binding evidence: weak
Native-like contacts: strong
Ligand efficiency: weak
Geometry reliability: low
Reason: geometry warning, clashes, strain 60.4 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 0 Clashes 24 Severe clashes 3
Final rank67.9264749606425Score7.53943
Inter norm-0.325994Intra norm0.455984
Top1000noExcludedyes
Contacts21H-bonds2
Artifact reasonexcluded; hard geometry fail; 2 severe clashes; 3 protein clashes; high raw intra
ResiduesA:ALA10;A:ARG29;A:ASN65;A:GLN36;A:GLU31;A:ILE61;A:ILE8;A:LEU23;A:LEU68;A:LYS64;A:LYS69;A:NAP201;A:PHE32;A:PHE35;A:PRO27;A:PRO62;A:SER60;A:THR57;A:TYR122;A:VAL116;A:VAL9

Protein summary

200 residues
Protein targetT02Atoms3128
Residues200Chains2
Residue summaryLYS:374; LEU:361; GLU:240; VAL:224; ARG:192; PHE:180; ILE:171; PRO:168; ASN:140; SER:132; TYR:126; GLN:119; ASP:108; MET:102; THR:98; GLY:91

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name5SD8Contacts21
PoseOpen native poseH-bonds5
IFP residuesA:ALA10; A:ASN65; A:ASP22; A:GLN36; A:GLU31; A:GLY117; A:GLY21; A:ILE61; A:ILE8; A:LEU23; A:LEU68; A:NAP201; A:PHE32; A:PHE35; A:PRO62; A:SER60; A:THR137; A:THR57; A:TYR122; A:VAL116; A:VAL9
Current overlap17Native recall0.81
Jaccard0.68RMSD-
H-bond strict0Strict recall0.00
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
371 12.07966259133659 -0.303826 12.7426 4 20 16 0.76 0.20 - no Open
364 10.700713840325998 -0.280321 -6.51466 5 17 14 0.67 0.00 - yes Open
374 10.74549312739154 -0.317175 -4.14822 4 20 16 0.76 0.00 - yes Open
370 58.499452820207246 -0.262113 6.60063 6 23 18 0.86 0.20 - yes Open
361 58.770600950025774 -0.389059 -0.519409 6 16 13 0.62 0.20 - yes Open
367 59.75725312034956 -0.339947 -20.3222 8 17 14 0.67 0.20 - yes Open
360 59.81246926598813 -0.421502 -0.157324 3 24 17 0.81 0.20 - yes Open
357 59.904211056420195 -0.338061 -12.2988 7 17 14 0.67 0.20 - yes Open
376 61.245461454346625 -0.232377 3.15961 3 19 15 0.71 0.20 - yes Open
366 61.31274073366522 -0.355319 -3.64314 3 22 18 0.86 0.20 - yes Open
356 61.40097881920791 -0.36586 -10.9336 5 19 13 0.62 0.20 - yes Open
359 61.48516176224802 -0.403851 -8.75094 4 20 17 0.81 0.20 - yes Open
377 61.51173990074728 -0.297892 -8.78728 6 20 17 0.81 0.20 - yes Open
368 61.7109151100752 -0.335379 20.4432 7 23 17 0.81 0.20 - yes Open
375 62.124241444784914 -0.312453 -7.35549 4 14 10 0.48 0.00 - yes Open
369 62.47825356073588 -0.310422 -3.44447 4 21 16 0.76 0.20 - yes Open
363 63.31816497785984 -0.278661 -14.8351 6 18 13 0.62 0.20 - yes Open
358 64.74757211702781 -0.328929 14.9784 4 24 18 0.86 0.20 - yes Open
362 64.80846384080228 -0.256903 11.2993 5 21 17 0.81 0.20 - yes Open
365 65.33790998459783 -0.29804 28.9055 8 20 15 0.71 0.20 - yes Open
373 65.54101327256443 -0.32434 -2.60468 4 24 20 0.95 0.20 - yes Open
372 67.9264749606425 -0.325994 7.53943 2 21 17 0.81 0.20 - yes Current

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score 7.539kcal/mol
Ligand efficiency (LE) 0.1300kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) 1.471
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 58HA

Physicochemical properties

Molecular weight 822.9Da
Lipinski: ≤ 500 Da
LogP (cLogP) 0.27
Lipinski: ≤ 5
Rotatable bonds 10

Conformational strain (MMFF94s)

Strain energy (ΔE) 60.43kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 132.97kcal/mol
Minimised FF energy 72.54kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.