FAIRMol

OHD_TB2022_21

Pose ID 3622 Compound 578 Pose 304

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.772 kcal/mol/HA) ✓ Good fit quality (FQ -7.91) ✓ Strong H-bond network (10 bonds) ✗ Very high strain energy (24.1 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-28.573
kcal/mol
LE
-0.772
kcal/mol/HA
Fit Quality
-7.91
FQ (Leeson)
HAC
37
heavy atoms
MW
495
Da
LogP
3.17
cLogP
Strain ΔE
24.1 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, protein contact clashes, strain 24.1 kcal/mol

Interaction summary

Collapsible panels
H-bonds 10 Hydrophobic 24 π–π 4 Clashes 3 Severe clashes 0
Final rank4.618637155274895Score-28.5727
Inter norm-0.803058Intra norm0.0308225
Top1000noExcludedno
Contacts21H-bonds10
Artifact reasongeometry warning; 17 clashes; 3 protein contact clashes; high strain Δ 29.1
ResiduesA:ALA32;A:ASP52;A:ILE45;A:LEU94;A:LYS57;A:MET53;A:NDP301;A:PHE55;A:PHE56;A:PHE91;A:PRO88;A:SER44;A:SER86;A:THR180;A:THR54;A:TYR162;A:TYR178;A:VAL156;A:VAL30;A:VAL31;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap18Native recall0.90
Jaccard0.78RMSD-
H-bond strict4Strict recall0.57
H-bond same residue+role4Role recall0.80
H-bond same residue4Residue recall0.80

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
304 4.618637155274895 -0.803058 -28.5727 10 21 18 0.90 0.80 - no Current
227 4.823152433370709 -1.14683 -33.4245 7 20 0 0.00 0.00 - no Open
197 4.832421871029605 -0.633104 -20.201 4 17 0 0.00 0.00 - no Open
197 5.121721553289744 -0.649791 -18.9976 4 19 1 0.05 0.00 - no Open
207 5.142565175193588 -0.544743 -15.1314 4 16 0 0.00 0.00 - no Open
204 5.158661328225735 -1.11363 -36.2955 9 21 0 0.00 0.00 - no Open
228 5.235002079928121 -0.934212 -30.9377 5 18 0 0.00 0.00 - no Open
178 6.391970965155197 -0.611124 -18.0149 5 20 0 0.00 0.00 - no Open
251 7.1983409405374275 -0.537335 -16.6239 3 15 0 0.00 0.00 - no Open
196 7.475422160355843 -0.717527 -22.2933 7 21 0 0.00 0.00 - no Open
302 7.904069850528994 -0.906033 -25.6212 7 24 19 0.95 0.20 - no Open
226 7.351286921462457 -1.00732 -33.1264 4 21 0 0.00 0.00 - yes Open
201 7.373429719771494 -1.03536 -33.075 7 20 0 0.00 0.00 - yes Open
202 7.880459488386842 -1.14596 -33.7036 7 21 0 0.00 0.00 - yes Open
252 7.895986744012289 -0.711971 -23.6267 8 16 0 0.00 0.00 - yes Open
203 8.070886547796118 -1.0222 -30.5113 5 19 0 0.00 0.00 - yes Open
229 8.291873648095919 -1.0842 -35.0367 11 20 0 0.00 0.00 - yes Open
303 8.45361427934496 -0.798578 -23.1576 8 22 19 0.95 0.40 - yes Open
205 8.645287298237387 -0.511082 -14.8838 3 14 0 0.00 0.00 - yes Open
176 9.267056293692587 -0.607051 -16.0283 5 15 0 0.00 0.00 - yes Open
305 10.742603935914689 -0.965604 -29.7543 10 21 17 0.85 0.60 - yes Open
177 10.93161836458181 -0.600757 -17.5629 5 13 0 0.00 0.00 - yes Open
206 11.386361520289974 -0.546086 -14.5867 6 14 0 0.00 0.00 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -28.573kcal/mol
Ligand efficiency (LE) -0.7722kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -7.906
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 37HA

Physicochemical properties

Molecular weight 494.6Da
Lipinski: ≤ 500 Da
LogP (cLogP) 3.17
Lipinski: ≤ 5
Rotatable bonds 9

Conformational strain (MMFF94s)

Strain energy (ΔE) 24.09kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 105.83kcal/mol
Minimised FF energy 81.74kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.