FAIRMol

OSA_Lib_160

Pose ID 36193 Compound 2822 Pose 1552

DB Docking_panel_21Docking pose analysis is being read from this database.

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Weak Marginal quality. Consider only alongside better-scoring alternatives.
✓ Excellent LE (-0.748 kcal/mol/HA) ✓ Good fit quality (FQ -6.97) ✗ High strain energy (15.8 kcal/mol) ✗ Geometry warnings ✗ Protein contact clashes ℹ SASA not computed
Score
-20.185
kcal/mol
LE
-0.748
kcal/mol/HA
Fit Quality
-6.97
FQ (Leeson)
HAC
27
heavy atoms
MW
382
Da
LogP
4.03
cLogP
Strain ΔE
15.8 kcal/mol
SASA buried
computing…

Interaction summary

Collapsible panels
H-bonds 1 Hydrophobic 18 π–π 0 Clashes 3 Severe clashes 0
Final rank2.2314517834749723Score-20.1851
Inter norm-0.72759Intra norm-0.0200063
Top1000noExcludedno
Contacts15H-bonds1
Artifact reasongeometry warning; 9 clashes; 3 protein contact clashes; moderate strain Δ 14.8
ResiduesA:ALA209;A:ALA90;A:ASN208;A:ASN91;A:GLY214;A:GLY215;A:LEU73;A:LYS211;A:LYS89;A:MET70;A:PRO187;A:PRO212;A:PRO213;A:TYR210;A:VAL88

Protein summary

493 residues
Protein targetT16Atoms7551
Residues493Chains1
Residue summaryVAL:768; LYS:704; LEU:703; ILE:532; GLU:450; THR:434; ARG:408; PHE:400; ALA:390; ASN:350; PRO:350; GLY:336; SER:319; TYR:294; ASP:276; MET:221

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name6RB5Contacts12
PoseOpen native poseH-bonds0
IFP residuesA:ALA90; A:ARG74; A:GLY85; A:LEU73; A:LYS89; A:MET70; A:PHE83; A:PRO212; A:PRO213; A:SER86; A:SER87; A:VAL88
Current overlap7Native recall0.58
Jaccard0.35RMSD-
H-bond strict0Strict recall-
H-bond same residue+role0Role recall-
H-bond same residue0Residue recall-

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

No π–π interactions detected for this pose.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
1552 2.2314517834749723 -0.72759 -20.1851 1 15 7 0.58 - - no Current
1561 2.2706400610765347 -0.755459 -21.1223 2 11 6 0.50 - - no Open
1550 2.6041262670774237 -0.7254 -20.2409 2 13 8 0.67 - - no Open
1563 52.703432501874616 -0.801934 -21.6587 2 11 6 0.50 - - no Open
1553 52.946930303698224 -0.766517 -21.4584 2 12 7 0.58 - - no Open
1559 53.194394080244265 -0.816058 -22.4006 2 12 7 0.58 - - no Open
1551 53.60524633670407 -0.847689 -23.5582 3 12 7 0.58 - - no Open
1554 54.09757277343734 -0.795584 -20.8985 3 11 7 0.58 - - no Open
1555 54.68799709594195 -0.829556 -22.6204 2 13 7 0.58 - - no Open
1558 54.99234971783147 -0.751746 -19.6814 1 11 6 0.50 - - no Open
1560 53.93046912823212 -0.777814 -20.8651 2 14 7 0.58 - - yes Open
1562 54.26867329975677 -0.697259 -18.4947 2 11 9 0.75 - - yes Open
1556 54.295694584778886 -0.811744 -21.8369 2 13 8 0.67 - - yes Open
1548 54.32238023155886 -0.855975 -23.1027 3 12 8 0.67 - - yes Open
1557 55.03081381684143 -0.700252 -18.599 2 11 8 0.67 - - yes Open
1549 55.848667567373084 -0.799375 -21.048 3 11 7 0.58 - - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -20.185kcal/mol
Ligand efficiency (LE) -0.7476kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -6.975
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 27HA

Physicochemical properties

Molecular weight 382.0Da
Lipinski: ≤ 500 Da
LogP (cLogP) 4.03
Lipinski: ≤ 5
Rotatable bonds 3

Conformational strain (MMFF94s)

Strain energy (ΔE) 15.76kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 92.10kcal/mol
Minimised FF energy 76.34kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. It will be calculated automatically the next time this pose is loaded if a receptor PDB path is stored.