FAIRMol

OHD_TB2021_72

Pose ID 3598 Compound 751 Pose 280

DB Docking_panel_21Docking pose analysis is being read from this database.
Molecular metrics status: done
Cached molecular metrics are available for this pose.
Metrics cached · SASA missing

py3Dmol interaction viewer

Left: interactive complex viewer. Right: clickable PLIP-like interaction summary. Clicking an interaction thickens and highlights it in the 3D view.
Strict H-bonds Permissive H-bonds
Molecular report
Full metrics ↗
Reject Multiple quality flags — this pose should be deprioritised or discarded.
✓ Excellent LE (-0.433 kcal/mol/HA) ✓ Good fit quality (FQ -4.60) ✗ Very high strain energy (28.3 kcal/mol) ✗ Geometry warnings ℹ SASA not computed
Score
-18.625
kcal/mol
LE
-0.433
kcal/mol/HA
Fit Quality
-4.60
FQ (Leeson)
HAC
43
heavy atoms
MW
602
Da
LogP
5.07
cLogP
Strain ΔE
28.3 kcal/mol
SASA buried
computing…
Overall: Promising but geometrically suspicious
Binding evidence: strong
Native-like contacts: strong
Ligand efficiency: excellent
Geometry reliability: low
Reason: geometry warning, clashes, strain 28.3 kcal/mol

Interaction summary

Collapsible panels
H-bonds 2 Hydrophobic 24 π–π 3 Clashes 15 Severe clashes 2
Final rank59.500333992523814Score-18.6246
Inter norm-0.449625Intra norm0.0164942
Top1000noExcludedyes
Contacts19H-bonds2
Artifact reasonexcluded; geometry warning; 15 clashes; 2 protein clashes
ResiduesA:ARG48;A:ARG97;A:ILE45;A:LEU94;A:LYS57;A:LYS95;A:MET53;A:MET79;A:NDP301;A:PHE56;A:PHE91;A:PRO88;A:PRO93;A:SER86;A:THR54;A:THR83;A:TRP47;A:VAL156;A:VAL87

Protein summary

225 residues
Protein targetT03Atoms3428
Residues225Chains2
Residue summaryLEU:380; ARG:360; VAL:272; LYS:264; ALA:240; GLU:240; PRO:224; PHE:180; THR:154; ILE:152; SER:132; TYR:126; GLN:119; ASN:98; GLY:84; NDP:74

Native ligand reference

★ reference
Interaction fingerprint calculated directly from the uploaded native ligand without docking. Current H-bond mode: strict.
Name3CL9Contacts20
PoseOpen native poseH-bonds9
IFP residuesA:ALA32; A:ARG97; A:ASP52; A:ILE45; A:LEU94; A:LYS57; A:MET53; A:NDP301; A:PHE56; A:PHE91; A:PRO88; A:SER86; A:THR180; A:THR54; A:THR83; A:TYR162; A:VAL156; A:VAL30; A:VAL31; A:VAL87
Current overlap14Native recall0.70
Jaccard0.56RMSD-
H-bond strict2Strict recall0.29
H-bond same residue+role1Role recall0.20
H-bond same residue1Residue recall0.20

Hydrogen bonds

Mode: strict. Count shows atom-level H-bonds; unique residues in summary: 0.

π–π interactions

Native π–π recall is disabled because no explicit native π–π reference was stored.

Hydrophobic contacts

Clashes

All stored poses for this docking hit

PoseFinal rankInter normScoreHBContactsNative overlapNative recallHB role recallRMSDExcluded
183 5.387499765091102 -0.445838 -21.9402 1 18 0 0.00 0.00 - no Open
177 6.419617103379667 -0.428919 -16.8141 3 17 0 0.00 0.00 - no Open
179 6.857077245144877 -0.491315 -18.6128 3 20 0 0.00 0.00 - no Open
287 10.773278844478433 -0.547189 -19.5005 4 16 12 0.60 0.20 - no Open
180 57.434866999748294 -0.422485 -17.9876 2 18 0 0.00 0.00 - no Open
285 10.220014194693826 -0.485907 -16.9188 2 14 12 0.60 0.20 - yes Open
284 10.262117288182628 -0.697159 -27.8016 3 18 14 0.70 0.20 - yes Open
178 57.902131558057945 -0.467181 -15.7119 6 19 0 0.00 0.00 - yes Open
182 58.41845885231413 -0.338607 -13.9156 3 17 0 0.00 0.00 - yes Open
176 58.905503850093744 -0.511703 -18.8363 2 18 0 0.00 0.00 - yes Open
181 59.27256112388008 -0.480704 -15.1847 1 17 0 0.00 0.00 - yes Open
280 59.500333992523814 -0.449625 -18.6246 2 19 14 0.70 0.20 - yes Current
283 59.715657803823824 -0.621342 -24.9099 3 18 16 0.80 0.20 - yes Open
281 60.75977422122872 -0.494045 -16.7876 2 17 12 0.60 0.20 - yes Open
282 61.8704921917718 -0.53851 -23.2696 2 19 13 0.65 0.20 - yes Open
286 63.8619445221105 -0.583095 -14.2429 2 19 15 0.75 0.20 - yes Open

Molecular metrics

FreeSASA-based burial, strain energy (MMFF94s), ligand efficiency and fit quality for this docking pose.
✓ Metrics available

Scoring & efficiency

Docking score -18.625kcal/mol
Ligand efficiency (LE) -0.4331kcal/mol/HA
Score / heavy atom count
Fit quality (FQ) -4.603
LE / (0.072 + 0.95/HAC) — Leeson & Springthorpe
Heavy atom count 43HA

Physicochemical properties

Molecular weight 601.7Da
Lipinski: ≤ 500 Da
LogP (cLogP) 5.07
Lipinski: ≤ 5
Rotatable bonds 13

Conformational strain (MMFF94s)

Strain energy (ΔE) 28.33kcal/mol
< 5 good · 5–10 marginal · > 10 problematic
Docked FF energy 82.14kcal/mol
Minimised FF energy 53.81kcal/mol

SASA & burial (FreeSASA)

not yet run
SASA has not been computed yet for this pose. Queue a background recompute to populate FreeSASA burial metrics without blocking the page.